Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VSLRVJBKRNJMHM
|
7.7 | IC50 | 2 | — | |
VXYDJXMHISGSDA
|
7.7 | Ki | 59 | — | |
WCCYEJYTLNWYCC
|
7.7 | IC50 | 9 | — | |
CVIBDXQYFNZNMA
|
7.7 | IC50 | 4 | — | |
DLPIYBKBHMZCJI
|
7.7 | IC50 | 12 | — | |
JLIQRHLZQGEBQQ
|
7.7 | IC50 | 3 | — | |
KYRQRRGDKAIFMA
|
7.7 | IC50 | 7 | — | |
NCBDOQFSGNRAHL
|
7.7 | IC50 | 6 | — | |
GIOKUJORFDKSSG
|
7.7 | IC50 | 7 | — | |
ASRWRMWLFZMROI
|
7.7 | IC50 | 6 | — | |
YPMOBRWHNOTUIL
|
7.7 | IC50 | 7 | — | |
ABTODZKWEKKTIC
|
7.6 | IC50 | 2 | — | |
AMHWMCSHBYIXCE
|
7.6 | IC50 | 3 | — | |
DTNFOGMAASDEQI
|
7.6 | IC50 | 5 | — | |
LVELIXLMLUGJEH
|
7.6 | IC50 | 4 | — | |
QNUKRWAIZMBVCU
|
7.6 | IC50 | 46 | — | |
LRJIEZPKWFBSEJ
|
7.6 | IC50 | 6 | — | |
PTAPBELLLOUDLL
|
7.6 | IC50 | 2 | — | |
QTHCAAFKVUWAFI
|
7.6 | IC50 | 23 | — | |
BIIVYFLTOXDAOV
|
7.6 | Ki | 31 | — | |
FLEAYYMORDPWAJ
|
7.6 | Ki | 90 | — | |
GFPGWHOCRYTVLL
|
7.6 | IC50 | 3 | — | |
IORBEYRNTKWGRM
|
7.6 | IC50 | 4 | — | |
MZWFSHNLGOBBSZ
|
7.6 | IC50 | 2 | — | |
OLVBAUVSICCWEJ
|
7.6 | Ki | 39 | — | |
POCZBHBFCIWCCV
|
7.6 | IC50 | 5 | — | |
QBKUOOQFSVMDPB
|
7.6 | Ki | 31 | — | |
QCOULMVHIHJKFY
|
7.6 | Ki | 14 | — | |
UZFPGFONVYFSRR
|
7.6 | Ki | 16 | — | |
VCTLOEWZYIGVBO
|
7.6 | IC50 | 12 | — | |
VMSMVRDDPGJMQF
|
7.6 | IC50 | 6 | — | |
YIAFFFACXVWBIZ
|
7.6 | IC50 | 4 | — | |
BZAMUGWDAXKCEU
|
7.6 | IC50 | 2 | — | |
UTBSBSOBZHXMHI
|
7.6 | IC50 | 15 | Yes | |
HHZHUPXWPPYGEU
|
7.6 | IC50 | 4 | — | |
YZSCPLGKKMSBMV
|
7.6 | IC50 | 10 | — | |
JKKUZTDMJDZHEB
|
7.6 | IC50 | 7 | — | |
AKDZNPFQMDRCMU
|
7.5 | IC50 | 7 | — | |
DSEWGOFKGFEZPE
|
7.5 | IC50 | 2 | — | |
IZOFFSRJFXHBHQ
|
7.5 | IC50 | 2 | — | |
LDLLFYVEDBJIIM
|
7.5 | IC50 | 2 | — | |
TYNCGTPANDPODX
|
7.5 | IC50 | 4 | — | |
ATBAETXFFCOZOY
|
7.5 | IC50 | 39 | — | |
DENJPOISBSHUGX
|
7.5 | IC50 | 2 | — | |
PGDIYOJSLLUWMQ
|
7.5 | Ki | 4 | — | |
POTKDJWRAMHALZ
|
7.5 | IC50 | 9 | — | |
SAKHMWHBWMDUMO
|
7.5 | IC50 | 7 | — | |
JRGMQQCQWFMKLA
|
7.5 | IC50 | 6 | — | |
HHZHUPXWPPYGEU
|
7.5 | IC50 | 4 | — | |
KRIWIRSMQRQYJG
|
7.5 | IC50 | 11 | — |