Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVKHEKZVCHMORX
|
7.9 | IC50 | 2 | — | |
YZXFATFOBBTPIG
|
7.9 | IC50 | 3 | — | |
CHTMRWQLNNRRFJ
|
7.9 | Ki | 70 | — | |
DQPYZHUAILXFJI
|
7.9 | Ki | 27 | — | |
HZPACYSNLOCDLW
|
7.9 | Ki | 48 | — | |
KAZJIBCOYQRDGG
|
7.9 | Ki | 16 | — | |
NJPWCTYVEJIQBM
|
7.9 | Ki | 72 | — | |
NLUPJKQOKWBWFC
|
7.9 | Ki | 69 | — | |
RYYNGWLOYLRZLK
|
7.9 | Ki | 104 | — | |
SBFPHSVZEXSHTL
|
7.9 | Ki | 62 | — | |
SLKCVFPEQGHNSI
|
7.9 | Ki | 29 | — | |
ZGZVRPRSFXRGCF
|
7.9 | Ki | 76 | — | |
BBSYDDJGTACDNC
|
7.9 | IC50 | 3 | — | |
JPWSUSDWOYHFRI
|
7.9 | IC50 | 3 | — | |
ORKSQVXJLGIROJ
|
7.9 | IC50 | 4 | — | |
SYKKXAMILDNUNO
|
7.9 | IC50 | 4 | — | |
TWGKEDPPHSZRCI
|
7.9 | IC50 | 3 | — | |
DIWRYQKRDLUVMY
|
7.8 | IC50 | 2 | — | |
NPXTWLXCVUMFMN
|
7.8 | IC50 | 2 | — | |
PEMNVVTZKGRLSX
|
7.8 | IC50 | 7 | — | |
XKPZMRRASYJBKC
|
7.8 | IC50 | 7 | — | |
NBSJZWFDNFWQDN
|
7.8 | IC50 | 29 | — | |
FLIVKVQMXOAQAK
|
7.8 | IC50 | 15 | — | |
PCQPAKMJSYGXRE
|
7.8 | IC50 | 16 | — | |
VSFIYAYRTKMILQ
|
7.8 | IC50 | 2 | — | |
VUKGJVXJRDQYFA
|
7.8 | IC50 | 9 | — | |
KGJVKYSVVOQPDL
|
7.8 | IC50 | 13 | — | |
RHWIDIZNQRAAIU
|
7.8 | IC50 | 7 | — | |
DSHAIQLEQCKJIR
|
7.8 | IC50 | 7 | — | |
DVBHEDLDLJERFO
|
7.8 | Ki | 9 | — | |
HRDHSMRDGZGSBV
|
7.8 | IC50 | 3 | — | |
KDJGCVHPUMHUOL
|
7.8 | Ki | 11 | — | |
NFTJDXGFOUFNKG
|
7.8 | IC50 | 16 | — | |
QHNBDDABNDUESC
|
7.8 | IC50 | 3 | — | |
VWVYILCFSYNJHF
|
7.8 | Ki | 49 | — | |
FKAJEPVSQITQLJ
|
7.8 | IC50 | 15 | — | |
JZBRRQXXXSBXIS
|
7.8 | IC50 | 3 | — | |
SVBJNUDKKXGVHI
|
7.8 | IC50 | 5 | — | |
GANPMWWREYHGFT
|
7.8 | IC50 | 2 | — | |
MNKJDIFJOOLBQY
|
7.8 | IC50 | 3 | Yes | |
OVPNQJVDAFNBDN
|
7.8 | IC50 | 44 | Yes | |
WROPYEAREMSHKX
|
7.8 | IC50 | 2 | — | |
UVKLAINVJNUJNX
|
7.7 | IC50 | 10 | — | |
FZLZLIAOYSKHJC
|
7.7 | Ki | 11 | — | |
QNABDSWBQJKBHK
|
7.7 | IC50 | 45 | — | |
QYSWLINIQVNEDI
|
7.7 | IC50 | 4 | — | |
BOLOCLITWRGHFA
|
7.7 | IC50 | 6 | — | |
JJGSOVIZOMZMCS
|
7.7 | Ki | 35 | — | |
MDJCUXFFMNEBHG
|
7.7 | Ki | 13 | — | |
QATMNAAQTUISJK
|
7.7 | Ki | 13 | — |