Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BGYVWFZMYBWCNY
|
8.2 | Ki | 30 | — | |
LPILBMJJRGTKOQ
|
8.2 | Ki | 27 | — | |
PNYMCFQCHXFMCI
|
8.2 | IC50 | 2 | — | |
RVSKJUNTDGBSSS
|
8.2 | Ki | 25 | — | |
URNZTLZSAVLTIZ
|
8.2 | Ki | 26 | — | |
UZQXPHDZFUAMQS
|
8.2 | IC50 | 9 | — | |
XZONYYFHQICDAM
|
8.2 | Ki | 19 | — | |
YGKFZWJWKPZPQM
|
8.2 | Ki | 13 | — | |
ZGGIYFOLDBTZIL
|
8.2 | Ki | 27 | — | |
ZOJWMCDSTRTTOW
|
8.2 | IC50 | 2 | — | |
ADBUMAAMWCLEEI
|
8.2 | IC50 | 3 | — | |
GCYXEGSPUDSZJY
|
8.2 | IC50 | 17 | Yes | |
TYSWNLQZLBRNSE
|
8.2 | IC50 | 15 | — | |
IWSDTEGBQVXXON
|
8.1 | IC50 | 7 | — | |
JRNJNYBQQYBCLE
|
8.1 | Kd | 40 | Yes | |
UPQKBKLECVIXJR
|
8.1 | IC50 | 12 | — | |
GJOXRIYWDHESDF
|
8.1 | Ki | 27 | — | |
MVJMMLFMPWITEJ
|
8.1 | Ki | 110 | — | |
MYOLWRIHGCZZGE
|
8.1 | IC50 | 3 | — | |
OEPMKSHSBUZDIB
|
8.1 | IC50 | 2 | — | |
SHZPFCZPWGVEED
|
8.1 | Ki | 5 | — | |
XDNYSGYXQHZDEY
|
8.1 | IC50 | 3 | — | |
BNVJXUKXMSVXHJ
|
8.1 | IC50 | 2 | — | |
NCAQSQYHTSCOCV
|
8.1 | IC50 | 7 | — | |
CGKJOISVQXEPSG
|
8.1 | Ki | 9 | — | |
CQWBHMMWZICZRH
|
8.1 | IC50 | 10 | — | |
JWZMXYSZZSYDGV
|
8.1 | IC50 | 4 | — | |
PUVVKKBHOWNLRX
|
8.1 | IC50 | 2 | — | |
QPROYVRFSAMXGU
|
8.1 | IC50 | 3 | — | |
RVKNONNXSNALJV
|
8.1 | IC50 | 21 | — | |
DIASEXMEBNQQHZ
|
8.0 | IC50 | 13 | — | |
FFVIVTCGXATTRT
|
8.0 | IC50 | 4 | — | |
FUMCKNCUEAQHCV
|
8.0 | Ki | 103 | — | |
HJYHJYGXRBYDIG
|
8.0 | Ki | 23 | — | |
IYNDTACKOAXKBJ
|
8.0 | IC50 | 17 | — | |
OHPFNMNHNRGIBV
|
8.0 | IC50 | 2 | — | |
RSQPNXBTPUXMQN
|
8.0 | IC50 | 12 | — | |
UDFDIIVNIYWXDM
|
8.0 | Ki | 74 | — | |
UERCVNGBBXPFLH
|
8.0 | IC50 | 3 | — | |
VWACUNWBMWWMPJ
|
8.0 | Ki | 18 | — | |
XUFLBSMTYMFOQH
|
8.0 | Ki | 43 | — | |
IVPOEQUCSQIXKZ
|
8.0 | IC50 | 2 | — | |
NYCKILAUMKSIPT
|
8.0 | IC50 | 2 | — | |
ONPNTUDUPZVQGU
|
8.0 | IC50 | 2 | — | |
RWSCYFXGWJPUQX
|
8.0 | IC50 | 15 | — | |
UCAUIDINMHWADR
|
8.0 | IC50 | 4 | — | |
DCRIEDZZYPOGPK
|
8.0 | IC50 | 4 | — | |
AKGTYSYXMRZPBV
|
7.9 | IC50 | 9 | — | |
BBSNLVGUSKQSBU
|
7.9 | IC50 | 2 | — | |
FKAJEPVSQITQLJ
|
7.9 | IC50 | 15 | — |