Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RYUQDJFJKIZISW
|
6.1 | IC50 | 3 | — | |
VUZONKZVVRZLCR
|
6.1 | IC50 | 2 | — | |
XQZSGOBAYDQIAM
|
6.1 | IC50 | 3 | — | |
FIMQVQVVIKFGOF
|
6.1 | IC50 | 2 | — | |
QQUXFYAWXPMDOE
|
6.1 | IC50 | 31 | — | |
WYDFLIFFODTBQK
|
6.1 | IC50 | 2 | — | |
XIJUQWYHULMNJA
|
6.1 | IC50 | 2 | — | |
CDYAOTQTBFPDQP
|
6.1 | Ki | 2 | — | |
AWGZLVOZDDBKNB
|
6.0 | IC50 | 2 | — | |
GNMSKQTUYNKOHN
|
6.0 | IC50 | 2 | — | |
GYBKTTNXKZFJGM
|
6.0 | IC50 | 2 | — | |
HVIKNWLSYBPGOG
|
6.0 | IC50 | 8 | — | |
KZAAPNQFAUCLEX
|
6.0 | IC50 | 2 | — | |
NTHMDBBWWNTVAZ
|
6.0 | IC50 | 5 | — | |
RVNDFXJEYCICIV
|
6.0 | IC50 | 7 | — | |
SXIDCDVJCQQXAU
|
6.0 | IC50 | 2 | — | |
VGAXWFQZQONAPZ
|
6.0 | IC50 | 6 | — | |
VQDHETXWBIZKEQ
|
6.0 | IC50 | 3 | — | |
AHHFGEKSWVBFGA
|
6.0 | IC50 | 3 | — | |
CMWRPDHVGMHLSZ
|
6.0 | IC50 | 22 | — | |
FUMJKSZLZJFCAQ
|
6.0 | IC50 | 10 | — | |
KOZFSFOOLUUIGY
|
6.0 | Kd | 88 | Yes | |
XBPSBLTUCDXDKJ
|
6.0 | IC50 | 2 | — | |
ADGFCJBOYWVXMS
|
6.0 | IC50 | 2 | — | |
KAJXOWFGKYKMMZ
|
6.0 | IC50 | 26 | Yes | |
SJWUVVGOTOMGOH
|
6.0 | IC50 | 12 | — | |
UGZKQEQKKSESBU
|
6.0 | IC50 | 2 | — | |
VTDMTVMKVZXVSP
|
6.0 | IC50 | 4 | — | |
SJXZTTFVVYAFTL
|
6.0 | IC50 | 3 | — | |
BHGSKYNWCFIOHP
|
6.0 | Ki | 6 | — | |
BOVRWIMDXLBREC
|
6.0 | IC50 | 2 | — | |
BTHLNBWTKKAULX
|
6.0 | Ki | 16 | — | |
CHGLHVVJPSESHY
|
6.0 | IC50 | 4 | — | |
DCTYSUJRBPLBJT
|
6.0 | IC50 | 2 | — | |
DYNWEDRLLZIBOF
|
6.0 | Ki | 2 | — | |
FQEODTMNWMDUMD
|
6.0 | Ki | 25 | — | |
FTGAOPZDJRWUTG
|
6.0 | IC50 | 6 | — | |
GPHUVHHAWZLCIP
|
6.0 | IC50 | 4 | Yes | |
GXNCJJUXJCUZSD
|
6.0 | Ki | 2 | — | |
HGRMYMRCAGWXEQ
|
6.0 | IC50 | 6 | — | |
HSKVRPZJBMXFDX
|
6.0 | Ki | 20 | — | |
IUEBPIPDFMCSTP
|
6.0 | Ki | 29 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JLTBOCSFMNSLFH
|
6.0 | Ki | 9 | — | |
JMIIFJIJWDCOEP
|
6.0 | Ki | 15 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KPVCGFZWGAYXMV
|
6.0 | Ki | 7 | — | |
KRIUNPBAQZGFQA
|
6.0 | Ki | 76 | — | |
KTRGYJLQTZDGPX
|
6.0 | Ki | 9 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |