Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XIFOACAKNZNAPH
|
6.1 | IC50 | 3 | — | |
YINGJLOKKADRGU
|
6.1 | IC50 | 2 | — | |
DCHDOYXSTZNERE
|
6.1 | IC50 | 4 | — | |
FXBHGLNIIVGSSW
|
6.1 | IC50 | 2 | — | |
HUSMRQOIXJQIFL
|
6.1 | IC50 | 2 | — | |
OGVUFJDFXLGOBE
|
6.1 | IC50 | 2 | — | |
QHTWDGUIDGQFLU
|
6.1 | IC50 | 2 | — | |
VLRAQJXMEDKPDZ
|
6.1 | IC50 | 2 | — | |
VQUQBABVYFSBGV
|
6.1 | IC50 | 6 | — | |
YIPABWNHLAARFQ
|
6.1 | IC50 | 2 | — | |
DDQWMUPDCRTRHM
|
6.1 | IC50 | 2 | — | |
MEOSMYVZUOFNIN
|
6.1 | IC50 | 2 | — | |
MXABJFXBEHROMU
|
6.1 | IC50 | 2 | — | |
WWNYYKFWFGFOAR
|
6.1 | IC50 | 2 | — | |
XDWOJCBGKHQWNM
|
6.1 | IC50 | 2 | — | |
YJKLTUUIJIUZDP
|
6.1 | IC50 | 3 | — | |
BFTWSRLZLPPTHF
|
6.1 | IC50 | 2 | — | |
UFGCTWUIESUHQP
|
6.1 | IC50 | 7 | — | |
BNBWNJAILLASJW
|
6.1 | IC50 | 4 | — | |
DCPBIOSSTDLFHO
|
6.1 | IC50 | 3 | — | |
DTMZXHDQZQLTHA
|
6.1 | Ki | 21 | — | |
FAIHBCXQSBIRIL
|
6.1 | Ki | 22 | — | |
FGLPGUCHBHILNS
|
6.1 | Ki | 10 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
GLMWKEAUVZDGKE
|
6.1 | Ki | 23 | — | |
GVMDVMPNOAVKJR
|
6.1 | Ki | 26 | Yes | |
IJNGXROUMFEKDB
|
6.1 | Ki | 39 | — | |
IPZUHNOYKQXXBS
|
6.1 | Ki | 2 | — | |
MVAMOERRWMZNPJ
|
6.1 | Ki | 4 | — | |
NXLLJUGNPKTXQP
|
6.1 | IC50 | 2 | — | |
OILINXINODUEIB
|
6.1 | IC50 | 8 | — | |
OKMGGPIYQLLQFZ
|
6.1 | IC50 | 7 | — | |
PAHHKMMVQJCPJI
|
6.1 | IC50 | 8 | — | |
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
RKKIDHHGKNGTQI
|
6.1 | Ki | 28 | — | |
ULVWJFBHQIXEPE
|
6.1 | Ki | 10 | — | |
UQNNJYLAPYGZBD
|
6.1 | Ki | 28 | — | |
WAKGEHXTOOFEAE
|
6.1 | Ki | 27 | — | |
XGISVNPAZQTTIQ
|
6.1 | IC50 | 6 | — | |
ZETZOOFGTLYZGU
|
6.1 | IC50 | 4 | — | |
ZUHJPCPWABPZDY
|
6.1 | IC50 | 8 | — | |
DQVLNFBISYHATC
|
6.1 | IC50 | 2 | — | |
LZRHAZRGHSSHLR
|
6.1 | IC50 | 7 | — | |
NSCYRWPACRPZKJ
|
6.1 | IC50 | 2 | — | |
RURHVWQWTJYUPS
|
6.1 | IC50 | 9 | — | |
WLUFZZMAAGDSJH
|
6.1 | IC50 | 4 | — | |
YAWHDNMICKDBLA
|
6.1 | IC50 | 2 | — | |
AXHMASICYOQTRA
|
6.1 | IC50 | 2 | — | |
LSFAJUUYCKHDNF
|
6.1 | IC50 | 2 | — | |
PMQCIJDDBNRBBC
|
6.1 | IC50 | 7 | — |