Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJJXQANLOSWJLA
|
6.2 | IC50 | 2 | — | |
DMGFZUJASYYJLE
|
6.2 | IC50 | 2 | — | |
OJYINLHOEHUFHI
|
6.2 | IC50 | 7 | — | |
SZOYOCHRMSEEMG
|
6.2 | IC50 | 7 | — | |
UKVQMBJHWHGXOI
|
6.2 | IC50 | 4 | Yes | |
WTXITEQXXBKUKS
|
6.2 | IC50 | 2 | — | |
CGPYAXSYKQBYKJ
|
6.2 | IC50 | 12 | — | |
MILILGJHFMDHIJ
|
6.2 | IC50 | 7 | — | |
MSPSOTZCMILMJO
|
6.2 | IC50 | 2 | — | |
OBKVROGZKBOQSW
|
6.2 | IC50 | 3 | — | |
UERHZBRVJFZGJV
|
6.2 | IC50 | 2 | — | |
UGAJHTSPHACTLO
|
6.2 | IC50 | 3 | — | |
UGEYGBMCWLIANH
|
6.2 | IC50 | 5 | — | |
VHHGAKUAIUOQSN
|
6.2 | IC50 | 2 | — | |
XZWSEBMTGSWQPC
|
6.2 | IC50 | 3 | — | |
YWUCEUICJFTKSJ
|
6.2 | IC50 | 3 | — | |
BTNSFEKKJRYFMD
|
6.2 | IC50 | 2 | — | |
CQLFRGIYOHYSJV
|
6.2 | IC50 | 7 | — | |
GYDXFTMHNUETBY
|
6.2 | IC50 | 5 | — | |
JQHYOJSXOWRHFO
|
6.2 | IC50 | 2 | — | |
KAGWQDFFFLWBFD
|
6.2 | IC50 | 8 | — | |
LETKAPAOLTWAHA
|
6.2 | IC50 | 2 | — | |
OIZWDVROSJCXER
|
6.2 | IC50 | 2 | — | |
OQUWTJLQOZIRFA
|
6.2 | IC50 | 8 | — | |
QMUKOEKTUBVPFU
|
6.2 | IC50 | 12 | — | |
QSZVFNDCIXARSO
|
6.2 | IC50 | 2 | — | |
VXUBVHRAMUWWBJ
|
6.2 | IC50 | 3 | — | |
XGRKGHCNVDZQGD
|
6.2 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
6.2 | Ki | 55 | — | |
BMKHCMLGQGVJTF
|
6.2 | Ki | 2 | — | |
DLIQZVFUDBYCQV
|
6.2 | IC50 | 2 | — | |
DYSRECIVMDGUQU
|
6.2 | Ki | 29 | — | |
FTAZWKPZLCOOEF
|
6.2 | IC50 | 2 | — | |
HGUSGBLHYRXWQF
|
6.2 | IC50 | 2 | — | |
IBBLSZHHKAUMBJ
|
6.2 | IC50 | 2 | — | |
KIJRIJFRVAOZCO
|
6.2 | IC50 | 2 | — | |
KKERJEDNLKDSOA
|
6.2 | IC50 | 2 | — | |
RGOPHVZLEMGMBZ
|
6.2 | Ki | 20 | — | |
SKGANWVAQNEQFN
|
6.2 | IC50 | 7 | — | |
SPOBBSBKXJKGBG
|
6.2 | Ki | 16 | — | |
UMYBAQLXZPEUQW
|
6.2 | Ki | 15 | — | |
WJRRGYBTGDJBFX
|
6.2 | Kd | 16 | Yes | |
XSRHBCYNCKAFKS
|
6.2 | Ki | 45 | — | |
YDOPLCNFRXOHCC
|
6.2 | Ki | 28 | — | |
BUVYKPYRCDJPQC
|
6.2 | IC50 | 2 | — | |
DHQGAPUQPLGEAC
|
6.2 | IC50 | 2 | — | |
DVGFYDFAEJURIW
|
6.2 | IC50 | 2 | — | |
FDGPWUHPMLUCBC
|
6.2 | IC50 | 2 | — | |
FNPZUYFPPNXJHB
|
6.2 | IC50 | 2 | — | |
HJQYXADEUQKZTJ
|
6.2 | IC50 | 2 | — |