Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QCPPFYUIILHREE
|
6.3 | IC50 | 2 | — | |
QZZHYZMBAUORBR
|
6.3 | IC50 | 3 | — | |
SDTHQOXRWZXTJF
|
6.3 | Ki | 16 | — | |
UTFXYGYVDDLJER
|
6.3 | Ki | 36 | — | |
UWZGPKLUCAHSOA
|
6.3 | IC50 | 5 | — | |
WMFVCLKZYKMDNK
|
6.3 | IC50 | 8 | — | |
CURXWONZHCZVOV
|
6.3 | IC50 | 5 | — | |
HQHSJJZIICGOIX
|
6.3 | IC50 | 8 | Yes | |
MUOKSQABCJCOPU
|
6.3 | Kd | 36 | — | |
PMXIKEQFDKDKSV
|
6.3 | IC50 | 2 | — | |
YALCKKGYRIHSMK
|
6.3 | IC50 | 2 | — | |
CKZIROWEZRCNOG
|
6.3 | IC50 | 2 | — | |
CVIZQDCZKWMREN
|
6.3 | IC50 | 2 | — | |
GGRHZNARBZKGTM
|
6.3 | IC50 | 2 | — | |
QQGVIAUMZWZUCW
|
6.3 | IC50 | 2 | — | |
UCJUQIKMOSVOJR
|
6.3 | IC50 | 2 | — | |
WKMWVRQSEXHGRD
|
6.3 | IC50 | 2 | — | |
AXWXMUIURGSJKE
|
6.3 | IC50 | 2 | — | |
CZANBJDHIJIHIW
|
6.3 | IC50 | 2 | — | |
FXLYXLFCTRGBDR
|
6.3 | IC50 | 2 | — | |
IJRXBGCUJWLVIO
|
6.3 | IC50 | 2 | — | |
IPVQXNIQUBCWRM
|
6.3 | IC50 | 2 | — | |
KCZYNJRAESMWAS
|
6.3 | IC50 | 2 | — | |
MFOAVBMJEANRPV
|
6.3 | IC50 | 2 | — | |
RAGGWBYDCQVJOC
|
6.3 | IC50 | 2 | — | |
ZDEBEWQYXJZQRS
|
6.3 | IC50 | 12 | — | |
ZWHTWAOLEGXRTP
|
6.3 | IC50 | 5 | — | |
DZLPPYFWEOZTEY
|
6.3 | IC50 | 3 | Yes | |
GKGZVFYMXSXLJJ
|
6.3 | IC50 | 2 | — | |
GSRHVOVIIWBRTN
|
6.3 | IC50 | 5 | — | |
JWLDHBNDOXSDBJ
|
6.3 | IC50 | 2 | — | |
LNDFIOHOUFFVLV
|
6.3 | IC50 | 2 | — | |
LZXYKKBAENJHCB
|
6.3 | IC50 | 2 | — | |
OBJNFLYHUXWUPF
|
6.3 | IC50 | 17 | — | |
SEWDWDRTQDIYJY
|
6.3 | IC50 | 2 | — | |
VCJRZTNERSUVFX
|
6.3 | IC50 | 2 | — | |
YBVSJBLXFZBKSU
|
6.3 | IC50 | 3 | — | |
KHGRVJUNFQKXRK
|
6.2 | IC50 | 2 | — | |
MNIRNNIUJSQGGD
|
6.2 | IC50 | 2 | — | |
OILWAOBAXWZBEF
|
6.2 | IC50 | 2 | — | |
PEIFTZAJJRCFLD
|
6.2 | IC50 | 2 | — | |
URTLBRVRTJEHIC
|
6.2 | IC50 | 2 | — | |
WGEJYGMWZJKLCB
|
6.2 | IC50 | 2 | — | |
BMENILZQTOWPIT
|
6.2 | IC50 | 2 | — | |
COTHGGLFZPNMEM
|
6.2 | IC50 | 2 | — | |
ODDISVVZPVDGCA
|
6.2 | IC50 | 2 | — | |
OGHRYYCQKDUEQB
|
6.2 | IC50 | 2 | — | |
QABMZNIZCUUCAD
|
6.2 | IC50 | 2 | — | |
SLNZFODXXSIZAB
|
6.2 | IC50 | 2 | — | |
ATRUDBHGBNHLHV
|
6.2 | IC50 | 2 | — |