Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBVOJALPYZEHOP
|
8.6 | Ki | 4 | — | |
XQVRYCHBRUAEMD
|
8.6 | IC50 | 2 | — | |
AAYPLLWGPJQWCC
|
8.5 | IC50 | 15 | Yes | |
CLCKDDAPJRHFEN
|
8.5 | IC50 | 9 | — | |
YRURITXEWXPMAI
|
8.5 | IC50 | 8 | Yes | |
YZVFJIYEYQIHIP
|
8.5 | IC50 | 15 | — | |
ZHMRPXZRUZLCNL
|
8.5 | IC50 | 8 | Yes | |
BXQKMGAINGBZAW
|
8.5 | IC50 | 11 | — | |
WDARYLSSWBWVCU
|
8.5 | Ki | 49 | — | |
DYHPOLTXTOPHPD
|
8.5 | IC50 | 2 | — | |
DZKMAWNYSJECKX
|
8.5 | IC50 | 12 | — | |
FGNHJXSBQQICEW
|
8.4 | Ki | 7 | — | |
IEGUVVCSOPRFMZ
|
8.4 | IC50 | 4 | — | |
HUHQPIYUPMEDGV
|
8.4 | IC50 | 2 | — | |
GNEARXSVRDSWKT
|
8.4 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
8.4 | IC50 | 408 | — | |
WADWOQCKXASRGQ
|
8.4 | IC50 | 4 | — | |
YRUAMADPOZOPBF
|
8.4 | IC50 | 7 | — | |
HKSZLNNOFSGOKW
|
8.4 | Ki | 118 | — | |
VASFNXBXECJRSY
|
8.4 | IC50 | 15 | — | |
VXBAJLGYBMTJCY
|
8.4 | IC50 | 34 | Yes | |
TVRXNAHDMVOXOV
|
8.4 | IC50 | 2 | — | |
KLJSQTWPBGAZHQ
|
8.4 | IC50 | 4 | — | |
DDPAPPCCQQJSAP
|
8.4 | IC50 | 9 | — | |
GFPPBUZAOLMYKX
|
8.4 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
8.4 | IC50 | 82 | — | |
NRKPJTBUHZKLGS
|
8.4 | Ki | 9 | — | |
YPJSFIQDRPQLPZ
|
8.4 | Ki | 9 | — | |
ZKCWYMOGNNWACW
|
8.4 | Ki | 4 | — | |
SZQYBGGKUBNKSZ
|
8.3 | IC50 | 5 | — | |
QYLYUTQSYHCBOD
|
8.3 | IC50 | 13 | — | |
BEJCLDKQCNVTQR
|
8.3 | Ki | 16 | — | |
BEMMPKXTCFGEAN
|
8.3 | IC50 | 5 | — | |
CJJMNECGBUPMAV
|
8.3 | IC50 | 8 | Yes | |
HUXYBQXJVXOMKX
|
8.3 | IC50 | 28 | — | |
JAPIBZGEANTMOW
|
8.3 | IC50 | 2 | — | |
MEWQZVRRNOXYMJ
|
8.3 | IC50 | 3 | — | |
MLSJNPCGOHGBCY
|
8.3 | IC50 | 3 | — | |
QBQOHKFVYIDSIJ
|
8.3 | IC50 | 6 | Yes | |
XFWUTMHVDGPWLH
|
8.3 | Ki | 75 | — | |
XLSYZSRXVVCHLS
|
8.3 | IC50 | 48 | — | |
FKAZCQZUYQPWFL
|
8.3 | IC50 | 2 | — | |
PUZNGRPTWFBCMK
|
8.2 | IC50 | 4 | — | |
CELCCCWTAADGDV
|
8.2 | IC50 | 15 | — | |
CSRROEXIZXVOPU
|
8.2 | IC50 | 4 | — | |
GIMRHZPQMMMJKH
|
8.2 | IC50 | 5 | — | |
KOLSEKSFVMGHDV
|
8.2 | IC50 | 12 | — | |
WESLFWSZUGLONY
|
8.2 | IC50 | 4 | — | |
YLWSVZLNZZVTSM
|
8.2 | IC50 | 15 | — | |
ZKDXRFMOHZVXSG
|
8.2 | IC50 | 13 | Yes |