Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FEGLECKDGAKPIQ
|
6.3 | IC50 | 2 | — | |
HDWRLGLOZANERH
|
6.3 | IC50 | 2 | — | |
HREZNQKDYUBSEM
|
6.3 | IC50 | 2 | — | |
HZGBRSQWJMBAES
|
6.3 | IC50 | 2 | — | |
JHRGHRGZTPOKRS
|
6.3 | IC50 | 2 | — | |
JNAXLMLGCBKAHT
|
6.3 | IC50 | 2 | — | |
MTNXGQDKMNFXJN
|
6.3 | IC50 | 2 | — | |
MYEGSPDGKBBLMH
|
6.3 | IC50 | 2 | — | |
NHUPUIRYSOEJFS
|
6.3 | IC50 | 2 | — | |
PVCCOICYYRDEPR
|
6.3 | IC50 | 2 | — | |
QFWXDBFSODFQPQ
|
6.3 | IC50 | 2 | — | |
RKWJSIVDWMXRNX
|
6.3 | IC50 | 2 | — | |
UFFCDEYMJYOOBI
|
6.3 | IC50 | 2 | — | |
UZIATSFXNVOVFE
|
6.3 | IC50 | 9 | — | |
VXYUPNCIMSOMFP
|
6.3 | IC50 | 2 | — | |
WTQKAOWVYODESZ
|
6.3 | IC50 | 2 | — | |
XNGZBKDVNBKPPD
|
6.3 | IC50 | 2 | — | |
ZGUKJPFTXCBWEJ
|
6.3 | IC50 | 2 | — | |
ZINPRHUOIGOZQZ
|
6.3 | IC50 | 2 | — | |
BOLOCLITWRGHFA
|
6.3 | IC50 | 5 | — | |
IVVIGIZSDTXDPN
|
6.3 | IC50 | 2 | — | |
LOFJRBSELKOTCG
|
6.3 | IC50 | 2 | — | |
NIOMALOJSIWPOB
|
6.3 | IC50 | 2 | — | |
OHARPIGKJAKOCM
|
6.3 | IC50 | 8 | — | |
OPSMLSVVHFWNNL
|
6.3 | IC50 | 2 | — | |
OPTXARRVRTXSQW
|
6.3 | IC50 | 2 | — | |
OWXORKPNCHJYOF
|
6.3 | IC50 | 17 | Yes | |
RYYNGWLOYLRZLK
|
6.3 | Kd | 45 | — | |
TXZCKJRNVSDDBF
|
6.3 | IC50 | 2 | — | |
VRSPGAKIMFTTJM
|
6.3 | IC50 | 2 | — | |
YROUADHZQZZZOP
|
6.3 | IC50 | 2 | — | |
FDDOKWKRYTUZJI
|
6.3 | IC50 | 2 | — | |
QHGYHFWTKKIXPB
|
6.3 | IC50 | 2 | — | |
UPFXMAHIEBOWOE
|
6.3 | IC50 | 2 | — | |
ANVTUJNDAMJQMR
|
6.3 | IC50 | 2 | — | |
AUBBSDZYWJYPEN
|
6.3 | IC50 | 2 | — | |
BNBWNJAILLASJW
|
6.3 | IC50 | 4 | — | |
DFMCXVONDDGQIY
|
6.3 | Ki | 66 | — | |
DUZUWJBAONJCTE
|
6.3 | IC50 | 7 | — | |
FSARIOOLDAHDFL
|
6.3 | IC50 | 5 | — | |
GKODJBVKKLQMEY
|
6.3 | Ki | 10 | — | |
HQRGSBHKKKWODU
|
6.3 | IC50 | 5 | — | |
IMMZLRQJNZSTTE
|
6.3 | Ki | 15 | — | |
KCKXYZOBGBJZEG
|
6.3 | Ki | 36 | — | |
MCKPYPWHBUXLEZ
|
6.3 | Ki | 21 | — | |
NIIWDVWAZLNFPB
|
6.3 | IC50 | 2 | — | |
OIDZQWOKVFYZSD
|
6.3 | Ki | 8 | — | |
PPWQAOVOMPHJDZ
|
6.3 | IC50 | 5 | — | |
PROLIXHVRCJEFH
|
6.3 | Ki | 46 | — | |
PTXLIQGTDWMAAF
|
6.3 | IC50 | 5 | — |