Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NWOJZWHRHFCZST
|
6.4 | IC50 | 2 | — | |
PGPHHJBZEGSUNE
|
6.4 | IC50 | 21 | — | |
UIARLYUEJFELEN
|
6.4 | Kd | 289 | Yes | |
ZXDDMQWKXGSSLJ
|
6.4 | IC50 | 3 | — | |
CJJQIFCAGQGNDS
|
6.4 | IC50 | 2 | — | |
FWWFACDHZONWBS
|
6.4 | IC50 | 2 | — | |
GMHOTJPHDRSKTA
|
6.4 | IC50 | 4 | — | |
HOSGYLWDAJEBNB
|
6.4 | IC50 | 3 | — | |
KLEHZMSJCLNMTM
|
6.4 | IC50 | 2 | — | |
KQINIHDQMUXUNU
|
6.4 | IC50 | 7 | — | |
LXFHUMQORRAHPG
|
6.4 | IC50 | 2 | — | |
NDIUYMHNCUTVGE
|
6.4 | Ki | 25 | — | |
NQVIIUBWMBHLOZ
|
6.4 | IC50 | 9 | Yes | |
QHTJZFWEQYRYQE
|
6.4 | IC50 | 9 | — | |
RIEOUYDQDXLXNM
|
6.4 | IC50 | 2 | — | |
XINSIGOHVDSHMB
|
6.4 | IC50 | 2 | — | |
XSEPRLAMFBFHKQ
|
6.4 | IC50 | 2 | — | |
YZDMOZWWDJLHJB
|
6.4 | IC50 | 2 | — | |
CIFXBRUONHOMEE
|
6.4 | IC50 | 2 | — | |
FFDUSKJJQOASLK
|
6.4 | IC50 | 2 | — | |
GDNYJRCASIYXQQ
|
6.4 | IC50 | 2 | — | |
RUELYCLIURLCMC
|
6.4 | IC50 | 2 | — | |
RVTOIQOTZUKDTE
|
6.4 | IC50 | 7 | — | |
XXOSKHOFQSTKGG
|
6.4 | IC50 | 2 | — | |
CGDONUPSODBGTG
|
6.4 | IC50 | 2 | — | |
FMRIUIOLOAMIMN
|
6.4 | IC50 | 2 | — | |
JGXGEUCTMRKONU
|
6.4 | IC50 | 2 | — | |
KSPPPMUBZRREPP
|
6.4 | IC50 | 2 | — | |
LJWNCENKRCHNIH
|
6.4 | IC50 | 2 | — | |
MYKPWRUVZULGRH
|
6.4 | IC50 | 4 | — | |
NVTINYQXFHNHIJ
|
6.4 | IC50 | 4 | — | |
QDSRRVVXMVAXFW
|
6.4 | IC50 | 2 | — | |
SBQWVNFVARONDG
|
6.4 | IC50 | 2 | — | |
UVJQEKJPAVSBTA
|
6.4 | IC50 | 8 | — | |
FMEOMSYWMHIHTC
|
6.3 | IC50 | 2 | — | |
SQUXCSCQSWIOMD
|
6.3 | IC50 | 2 | — | |
ABZXRAQIVBXXPG
|
6.3 | IC50 | 3 | — | |
CGTXNUPYOHWTIB
|
6.3 | IC50 | 2 | — | |
DKXHSOUZPMHNIZ
|
6.3 | IC50 | 51 | Yes | |
GDNSQFYYOWJJFA
|
6.3 | IC50 | 2 | — | |
GWVIPPFFKAJRAS
|
6.3 | IC50 | 2 | — | |
HGLXMQVHFPPLAQ
|
6.3 | IC50 | 2 | — | |
MCLSFEBANGIFLQ
|
6.3 | IC50 | 2 | — | |
OBJKGCVTCMNBNC
|
6.3 | IC50 | 2 | — | |
QJXQNPUOXVXJKG
|
6.3 | IC50 | 2 | — | |
UHOPJKMQVDXYAV
|
6.3 | IC50 | 8 | — | |
ANHREWRCDHYDAG
|
6.3 | IC50 | 2 | — | |
APSMLYMGHNAQFU
|
6.3 | IC50 | 2 | — | |
DROYSTDUOMEFHS
|
6.3 | IC50 | 2 | — | |
DWJHXWVIKXENPB
|
6.3 | IC50 | 2 | — |