Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JJPAZEYTVSKMAD
|
6.4 | IC50 | 3 | — | |
MFIOEGZMANTECR
|
6.4 | IC50 | 2 | — | |
CWLMDLJQXOAVGI
|
6.4 | IC50 | 2 | — | |
GLPRZGTYPDHMRV
|
6.4 | IC50 | 2 | — | |
LPGJKZZMPXMBSF
|
6.4 | IC50 | 2 | — | |
LVXRFLQOPGSERY
|
6.4 | IC50 | 2 | — | |
WHNSGFXLCCFUNW
|
6.4 | IC50 | 2 | — | |
AINKQRBPBUTJRM
|
6.4 | IC50 | 5 | — | |
CXBHZMHGPNBDBJ
|
6.4 | IC50 | 3 | — | |
DBAYOMQZYDSJKV
|
6.4 | IC50 | 2 | — | |
DURPLUQLWLERHZ
|
6.4 | IC50 | 2 | — | |
KHPWKCOFVQNLDH
|
6.4 | IC50 | 2 | — | |
MVCOAUNKQVWQHZ
|
6.4 | Kd | 54 | Yes | |
RTECFPIGBVOCPH
|
6.4 | IC50 | 2 | — | |
VAGFVMVMAWDHLF
|
6.4 | IC50 | 2 | — | |
YJGWBXGIQWQMLW
|
6.4 | IC50 | 2 | — | |
ZLIAMJQWKIUHTK
|
6.4 | IC50 | 2 | — | |
AEZICWXXUCODMN
|
6.4 | Ki | 8 | — | |
ATFBEKGTULYWDD
|
6.4 | IC50 | 5 | — | |
AWEGSLJDAPXFHZ
|
6.4 | IC50 | 2 | — | |
BLTVBQXJFVRPFK
|
6.4 | Ki | 7 | — | |
CMVVZTDBEHPABJ
|
6.4 | IC50 | 2 | — | |
DPEXRCOBPACFOO
|
6.4 | Ki | 36 | — | |
DWHVZCLBMTZRQM
|
6.4 | IC50 | 6 | — | |
FINBCMQWNUIQOI
|
6.4 | IC50 | 2 | — | |
FVOYXCNJIASCPE
|
6.4 | IC50 | 5 | — | |
GWXPHWSUMLUDPO
|
6.4 | Ki | 11 | — | |
HDRLAVNNWSHSOA
|
6.4 | Ki | 19 | — | |
HEUSUIRCBWROMH
|
6.4 | Ki | 64 | — | |
HNGSMPZLGYDZOV
|
6.4 | IC50 | 4 | — | |
IPTSYCYNQJITNJ
|
6.4 | Ki | 12 | — | |
IZRCBCKFMRACRK
|
6.4 | IC50 | 3 | — | |
LACOMQAWPSFXQC
|
6.4 | Ki | 27 | — | |
LDHYCINFJPCBRY
|
6.4 | Ki | 9 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
OEKYVFZKBRIDJO
|
6.4 | Ki | 12 | — | |
OFGKHGRQQKNHAV
|
6.4 | Ki | 5 | — | |
OHLKBSAOSZPTFS
|
6.4 | Ki | 9 | Yes | |
PUYIXDDMOUMMRR
|
6.4 | Ki | 27 | — | |
VGGWPBMWNFKYBD
|
6.4 | IC50 | 2 | — | |
WCVWDOVRLYUENM
|
6.4 | IC50 | 2 | — | |
WDIWPOWDVBIWKH
|
6.4 | IC50 | 2 | — | |
XSDJOIOVIMPMHD
|
6.4 | Ki | 44 | — | |
YTFZRCFWKAXGJK
|
6.4 | IC50 | 2 | — | |
YUOWJICKAJQZLS
|
6.4 | Ki | 35 | — | |
ZRQXCQXWTLVASO
|
6.4 | Ki | 36 | — | |
ZVWRFVCNQOECJS
|
6.4 | Ki | 71 | — | |
CLVVBNMTYMKNAP
|
6.4 | IC50 | 2 | — | |
KHKNDHVTUWWADD
|
6.4 | IC50 | 2 | — | |
MCCXYLHNBSSOCX
|
6.4 | IC50 | 2 | — |