Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LJJPTZDFLIRAPR
|
6.5 | IC50 | 2 | — | |
NKGLJTITEFZKAN
|
6.5 | Ki | 35 | — | |
OWDRQHVEJIYVOI
|
6.5 | Ki | 47 | — | |
PEXKNSGOEOREKM
|
6.5 | Ki | 13 | — | |
RKUKAACYUCUJEE
|
6.5 | Ki | 58 | — | |
SYLTYCLPHHSEIJ
|
6.5 | Ki | 27 | — | |
UYGYYOIUVFMGKQ
|
6.5 | Ki | 30 | — | |
WQFGNANQTYLQBP
|
6.5 | Ki | 16 | — | |
YDXQVABEPJBULM
|
6.5 | IC50 | 2 | — | |
YEKVTSRZMPLPFK
|
6.5 | Ki | 17 | — | |
KZZOJMWYRUFPAM
|
6.5 | IC50 | 3 | — | |
ZFUNUCBZILJMQN
|
6.5 | IC50 | 2 | — | |
DPDVVGCNUWGGRS
|
6.5 | IC50 | 10 | — | |
WMRINZZGUMOYEC
|
6.5 | IC50 | 4 | — | |
ZXLRQGOMWXZUTG
|
6.5 | IC50 | 2 | — | |
AHESLWPETCVNAQ
|
6.5 | IC50 | 2 | — | |
AMRDFGREILHODF
|
6.5 | IC50 | 2 | — | |
BSLQOWQMMZAVQV
|
6.5 | IC50 | 2 | — | |
GUDBDNYMUVSMPF
|
6.5 | IC50 | 2 | — | |
MHMOMLQYLUTCPX
|
6.5 | IC50 | 2 | — | |
NWPUNMUDGDUHRY
|
6.5 | IC50 | 2 | — | |
OUSFTKFNBAZUKL
|
6.5 | IC50 | 58 | Yes | |
OYRGDRUYBZTRNH
|
6.5 | IC50 | 2 | — | |
PMELCRDEYCUFNB
|
6.5 | IC50 | 5 | — | |
YHYSBRXGAHZSRA
|
6.5 | IC50 | 2 | — | |
IDLJEZYYKOQCEI
|
6.5 | IC50 | 2 | — | |
POFXHYGZNJNSKB
|
6.5 | IC50 | 2 | — | |
QEYLUQTVGIUEHV
|
6.5 | IC50 | 2 | — | |
DKQHTNGDIMXSBE
|
6.5 | IC50 | 2 | — | |
GWUNVPRNYCHCSX
|
6.5 | IC50 | 2 | — | |
IVSLHVMDZYSVFA
|
6.5 | IC50 | 3 | — | |
JVDVYWTYPYGQRD
|
6.5 | IC50 | 4 | — | |
NZWSUOOSFJXEEX
|
6.5 | IC50 | 2 | — | |
QKVOBTHWPHZLET
|
6.5 | IC50 | 3 | — | |
RAYGNBLIGRBJOW
|
6.5 | IC50 | 2 | — | |
SAAXYMYCHZMPBZ
|
6.5 | IC50 | 2 | — | |
UMDRMHHUBLRBRG
|
6.5 | IC50 | 2 | — | |
XRDCVWAKCKYRGJ
|
6.5 | IC50 | 2 | — | |
BUKNIOLWHFXEIG
|
6.4 | IC50 | 6 | — | |
FSDQIAXHAWLBNS
|
6.4 | IC50 | 2 | — | |
LYQFVXKEEXRKQE
|
6.4 | IC50 | 2 | — | |
NLJFBOXPANMGKW
|
6.4 | IC50 | 2 | — | |
OQUITAZKWLLMFX
|
6.4 | IC50 | 2 | — | |
QXOPSOWTTPTUKT
|
6.4 | IC50 | 2 | — | |
XFKCRUQXXNLAAT
|
6.4 | IC50 | 2 | — | |
ZSAQGXDSTQPMRV
|
6.4 | IC50 | 2 | — | |
ZZLGSHVSHBWPBE
|
6.4 | IC50 | 2 | — | |
BDGXXQSVGFGVOR
|
6.4 | IC50 | 2 | — | |
FQFGDUPFMGYOMB
|
6.4 | IC50 | 6 | — | |
IHMIELMZOYWQCJ
|
6.4 | IC50 | 2 | — |