Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MMAGRRZOKFIBFA
|
6.8 | IC50 | 2 | — | |
NGDQZHZQUZQYHB
|
6.8 | IC50 | 5 | — | |
OOYQNTZOMNZRSG
|
6.8 | IC50 | 8 | — | |
QOAWOYVJVKOWMX
|
6.8 | IC50 | 3 | — | |
RQUYLFVCZMFFCI
|
6.8 | IC50 | 4 | — | |
SMPPSGXPGZSJCP
|
6.8 | IC50 | 8 | — | |
CAFCQLWZFWROAD
|
6.7 | IC50 | 3 | — | |
KJLHEVSAJFFFGP
|
6.7 | IC50 | 3 | — | |
MOKFUAFGXXXFHR
|
6.7 | IC50 | 2 | — | |
DEYPVOVXSRFHNY
|
6.7 | IC50 | 2 | — | |
DYTKVFHLKPDNRW
|
6.7 | IC50 | 23 | Yes | |
IRKYBMOSIOKMFO
|
6.7 | IC50 | 2 | — | |
MMALMDVPDVEEIS
|
6.7 | IC50 | 2 | — | |
AJLCOLFEZAFAFY
|
6.7 | IC50 | 5 | — | |
BIUDJFOTQAVFMN
|
6.7 | IC50 | 9 | — | |
CZZCAOGIEGXMBZ
|
6.7 | IC50 | 10 | — | |
ONRSALYRJMUWEV
|
6.7 | IC50 | 2 | — | |
URBCMMCMDJBTCF
|
6.7 | IC50 | 2 | — | |
USIKZDCXQWHYCP
|
6.7 | IC50 | 2 | — | |
UZWDCWONPYILKI
|
6.7 | IC50 | 47 | — | |
YEWQGDMCRKBFBD
|
6.7 | IC50 | 3 | — | |
YGXHQYJKJUFSJI
|
6.7 | IC50 | 14 | — | |
FRCIRPZMZDFVMQ
|
6.7 | IC50 | 7 | — | |
JMDKLPDVAQXYMC
|
6.7 | IC50 | 2 | — | |
AOPRHEOJTUWSAR
|
6.7 | IC50 | 8 | — | |
BSFNGHCTZDCQBF
|
6.7 | Ki | 93 | — | |
BTIHMVBBUGXLCJ
|
6.7 | IC50 | 6 | — | |
BTIHMVBBUGXLCJ
|
6.7 | IC50 | 21 | Yes | |
DMGIJRJGSKIPRS
|
6.7 | IC50 | 2 | — | |
HPUUQGKVJFVXEY
|
6.7 | IC50 | 2 | — | |
HQRGSBHKKKWODU
|
6.7 | IC50 | 2 | — | |
KGCRKAITGGKXHI
|
6.7 | Ki | 5 | — | |
LAMQDGYKYXRPLW
|
6.7 | IC50 | 2 | — | |
LQYHWFFRRIMAPW
|
6.7 | IC50 | 5 | — | |
MPXAWSABMVLIBU
|
6.7 | IC50 | 6 | — | |
MRLQVJNPTNEGLQ
|
6.7 | IC50 | 2 | — | |
NCBDOQFSGNRAHL
|
6.7 | IC50 | 6 | — | |
NMOPSVILFGBLLC
|
6.7 | IC50 | 6 | — | |
NNOGQWYMWQTRCY
|
6.7 | IC50 | 2 | — | |
PRIGRJPRGZCFAS
|
6.7 | IC50 | 13 | Yes | |
PSCJSWRVCKUMSL
|
6.7 | Ki | 35 | — | |
PVKHDYBJGIJIAB
|
6.7 | IC50 | 2 | — | |
QBZJAAYUTYAIBM
|
6.7 | IC50 | 2 | — | |
QLUMKJWDOKCSJU
|
6.7 | IC50 | 3 | Yes | |
QZPFUALVXZAFDD
|
6.7 | Ki | 10 | — | |
RQJIDUOCLNMUHR
|
6.7 | Ki | 15 | — | |
RTDSHUGNRVXRHN
|
6.7 | Ki | 51 | — | |
SKKRZILJUKYLJS
|
6.7 | Ki | 25 | — | |
VDOHDCXDESGVKC
|
6.7 | IC50 | 8 | — | |
BBCSUMURJUYILA
|
6.7 | IC50 | 10 | — |