Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIQQNJQVGQVLBS
|
6.8 | IC50 | 2 | — | |
DFHRUTWHYJCTMH
|
6.8 | IC50 | 4 | — | |
GZKUIKKDBXPCIY
|
6.8 | IC50 | 13 | Yes | |
SDDXLJVXFBEYGV
|
6.8 | IC50 | 8 | — | |
SQVBZWHGFBQRIR
|
6.8 | IC50 | 5 | Yes | |
USBKPWRTJAXTBS
|
6.8 | IC50 | 16 | Yes | |
VTWWRKFUHCSCEW
|
6.8 | Kd | 19 | — | |
YFXBIIDXMTUIMX
|
6.8 | IC50 | 2 | — | |
NMFKDDRQSNVETB
|
6.8 | IC50 | 9 | Yes | |
VKLIPAKVEGHLJH
|
6.8 | IC50 | 2 | — | |
AKBYXQQHOAZMPQ
|
6.8 | IC50 | 3 | Yes | |
ASNDURJGUUDPHG
|
6.8 | Ki | 7 | — | |
ATBAETXFFCOZOY
|
6.8 | IC50 | 10 | — | |
BKQKPRMOYMYOAI
|
6.8 | IC50 | 2 | — | |
BQYDGSNDLAZAEW
|
6.8 | Ki | 13 | — | |
CVMAHPSTCONZBL
|
6.8 | IC50 | 2 | — | |
CXBZUFRMBVLFPL
|
6.8 | IC50 | 2 | — | |
DZIPQNPWTUXXSJ
|
6.8 | Ki | 18 | — | |
FTQZKKZJHPMZQD
|
6.8 | IC50 | 2 | — | |
GCBJDOWIQHMCMR
|
6.8 | Ki | 84 | — | |
IWPWKQLFCMXCMD
|
6.8 | Ki | 3 | — | |
JIPCPCOVWLXHPR
|
6.8 | IC50 | 2 | — | |
JJTYLBBKGQOISV
|
6.8 | Ki | 15 | — | |
JRNXAQINDCOHGS
|
6.8 | IC50 | 13 | — | |
LEBKMPSDNMCBGO
|
6.8 | IC50 | 2 | — | |
LNIDFQVRZCDVBI
|
6.8 | Ki | 16 | — | |
OAFSEOBYSMNKHG
|
6.8 | IC50 | 3 | — | |
ODNOTLMFNVWFTJ
|
6.8 | Ki | 11 | — | |
PEDNSWRLVHWPEG
|
6.8 | IC50 | 2 | — | |
SRONQUHCRFZABC
|
6.8 | Ki | 28 | — | |
UOVCGJXDGOGOCZ
|
6.8 | Ki | 59 | — | |
UQFRSHRWRKYNDE
|
6.8 | Ki | 17 | Yes | |
UWEHIBQNZMPNPF
|
6.8 | IC50 | 4 | — | |
XXSPHNFKLDJDAK
|
6.8 | Ki | 26 | — | |
AGLGNTHKUSBQJJ
|
6.8 | IC50 | 4 | — | |
IAQGXGNNLBONLG
|
6.8 | IC50 | 2 | — | |
GIONWDQPQBWBDK
|
6.8 | IC50 | 2 | — | |
ILSISQSFRSPFJR
|
6.8 | IC50 | 3 | — | |
SAOYLDFCVBRUJI
|
6.8 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.8 | IC50 | 82 | Yes | |
GGEWEQJWGGJUHO
|
6.8 | IC50 | 8 | Yes | |
LDICMBYRLCNQPK
|
6.8 | IC50 | 2 | — | |
TTYXOSBLVBJYMI
|
6.8 | IC50 | 2 | — | |
FONRCZUZCHXWBD
|
6.8 | IC50 | 8 | — | |
JRNXAQINDCOHGS
|
6.8 | IC50 | 15 | — | |
BTIHMVBBUGXLCJ
|
6.8 | IC50 | 7 | Yes | |
DRSBYEAJEUMMFA
|
6.8 | IC50 | 2 | — | |
FMLXCYYFKJXEAM
|
6.8 | IC50 | 2 | — | |
HDRGJVBNKICLJR
|
6.8 | IC50 | 6 | — | |
KBMRQCQCDYQDIH
|
6.8 | IC50 | 4 | — |