Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWGOHAYTCAXWHE
|
7.0 | IC50 | 2 | — | |
ABBWKPWBJVDHCD
|
6.9 | IC50 | 3 | — | |
RIGZCVNCFXYBEG
|
6.9 | IC50 | 11 | Yes | |
GJJRVWPGMNAXLZ
|
6.9 | IC50 | 3 | — | |
IAJGQMXAKJOLBA
|
6.9 | IC50 | 7 | — | |
NBOBLXOZHBALAX
|
6.9 | IC50 | 7 | — | |
NQORLXIULOFSFK
|
6.9 | IC50 | 2 | — | |
SIDJEVKSQLUEOQ
|
6.9 | IC50 | 2 | — | |
UJFAOQFICNRWOP
|
6.9 | IC50 | 4 | — | |
UQSJZZMWPULVAA
|
6.9 | IC50 | 2 | — | |
XBIUKPXUYROLSP
|
6.9 | IC50 | 2 | — | |
YQMRPYHUZUQSNB
|
6.9 | IC50 | 3 | Yes | |
BPNUQXPIQBZCMR
|
6.9 | Ki | 60 | — | |
CLEGDJQQHUTCOW
|
6.9 | Ki | 43 | — | |
CRKQBJZCCHKEGI
|
6.9 | Ki | 20 | — | |
GHPFQRTVUDXWCC
|
6.9 | Ki | 35 | — | |
HXESDBWWDYJEJQ
|
6.9 | Ki | 10 | — | |
JWQOJVOKBAAAAR
|
6.9 | Ki | 29 | — | |
NMHMCXTYPRADBA
|
6.9 | Ki | 20 | — | |
PLHUMPJXRHMFFR
|
6.9 | Ki | 28 | — | |
RSFBNWZRZYKDMI
|
6.9 | Ki | 4 | — | |
SEZFNTZQMWJIAI
|
6.9 | Ki | 22 | — | |
UJBJWYNPUOLFIZ
|
6.9 | Ki | 49 | — | |
WZBMMJKAHHOXRG
|
6.9 | Ki | 16 | — | |
ZGDYBJXDIXVTLV
|
6.9 | Ki | 54 | — | |
BYUPNMOFJSAIHN
|
6.9 | IC50 | 6 | — | |
JTXGWTJLZDKHJQ
|
6.9 | IC50 | 8 | — | |
MEJNYSXBLHEZDC
|
6.9 | IC50 | 2 | — | |
MWMTZLUYNDSKJP
|
6.9 | IC50 | 2 | — | |
NUYNGOGBVNFKBM
|
6.9 | IC50 | 2 | — | |
NXMIQKJGFTVADM
|
6.9 | IC50 | 4 | — | |
SQUNOCMDMIQIQK
|
6.9 | IC50 | 2 | — | |
FCLBVILBAPMKST
|
6.9 | IC50 | 13 | — | |
FMYDWZBWZKJPCK
|
6.9 | IC50 | 4 | — | |
LCDCVRYMEWMBEV
|
6.9 | IC50 | 5 | — | |
MUDAPTILNSVOOR
|
6.9 | IC50 | 2 | — | |
YQOZFMRCEONJEU
|
6.9 | IC50 | 13 | — | |
YRFOQHHFWYWAST
|
6.9 | IC50 | 22 | — | |
KHTQGWKOTJZKCD
|
6.9 | IC50 | 4 | — | |
ZNJIRQMCOQXGAV
|
6.9 | IC50 | 3 | — | |
KSIJGQVGLOGHKO
|
6.9 | IC50 | 2 | — | |
UEBSTEGTOAOQHT
|
6.9 | Ki | 4 | — | |
PBDNNWWYSHCMCH
|
6.8 | IC50 | 7 | — | |
QSQLSTWOUFBPKW
|
6.8 | IC50 | 4 | — | |
QXBKFUBBGBWPCJ
|
6.8 | IC50 | 8 | — | |
JMTLABPKNNCMFI
|
6.8 | IC50 | 2 | — | |
QIYXLIZWXGGKOO
|
6.8 | IC50 | 10 | — | |
RMQMCGSCLKFYRU
|
6.8 | IC50 | 2 | — | |
UCDVZAJSQRLZDD
|
6.8 | IC50 | 4 | — | |
AKKQLMPWVUMKJQ
|
6.8 | IC50 | 2 | — |