Target Details
| UniProt AC | Q00535 |
|---|---|
| Gene Symbol | CDK5 |
| Protein Name | Cyclin-dependent kinase 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,218
- Clinical molecules 62
- Avg pChEMBL 6.94
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (1,218)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SUEYATVNHWMTSO
|
7.1 | IC50 | 7 | — | |
ZPHBEDTYTQWLFC
|
7.1 | IC50 | 13 | — | |
LQHMJVOJVOLFTJ
|
7.1 | IC50 | 7 | — | |
PUXKEKPYASIYGT
|
7.1 | IC50 | 7 | — | |
WCEHIDWONYOKOJ
|
7.1 | IC50 | 3 | — | |
MZDKLVOWGIOKTN
|
7.1 | Kd | 80 | — | |
NXSJMRCTGYTSTK
|
7.1 | Kd | 200 | — | |
PFCAHEMJANLCHH
|
7.1 | IC50 | 2 | — | |
AREWHVALAPEARZ
|
7.0 | IC50 | 4 | — | |
IWXIAMLCFOOOMV
|
7.0 | IC50 | 8 | Yes | |
PRRNEKPNFWMEPT
|
7.0 | IC50 | 2 | — | |
UNLGUYJWTWLABD
|
7.0 | IC50 | 2 | — | |
VMSMVRDDPGJMQF
|
7.0 | IC50 | 5 | — | |
BNCYSCHURFNZGJ
|
7.0 | IC50 | 3 | — | |
CEIJSVLEARLWRF
|
7.0 | IC50 | 13 | — | |
CQVJGFKTRSGJHB
|
7.0 | Ki | 11 | — | |
UZUCFTPPULEGQO
|
7.0 | IC50 | 9 | — | |
WIAMCDYCLOMHKF
|
7.0 | IC50 | 6 | — | |
GJTRIRZIYRVGHG
|
7.0 | IC50 | 4 | — | |
QNWXRLPZIFMTBK
|
7.0 | IC50 | 12 | — | |
SVPUOZWGAJVQMQ
|
7.0 | IC50 | 2 | — | |
YWZXVOUKTPVGKU
|
7.0 | IC50 | 2 | — | |
ATGVCJYHNOSZEV
|
7.0 | Ki | 23 | — | |
CFBADDSSFSYJPF
|
7.0 | Ki | 23 | — | |
CHADTINFLWZSKR
|
7.0 | Ki | 26 | — | |
DMFMPEWLXMKYKK
|
7.0 | IC50 | 4 | — | |
FLHJZUQGFPJXRD
|
7.0 | Ki | 12 | — | |
FQCPPVRJPILDIK
|
7.0 | IC50 | 12 | — | |
HBDSHCUSXQATPO
|
7.0 | IC50 | 14 | Yes | |
HKECWLZKPZHUND
|
7.0 | IC50 | 8 | — | |
HWUAECSPBXTMLX
|
7.0 | IC50 | 2 | — | |
JSJVSQMHVJPNON
|
7.0 | IC50 | 5 | — | |
LRINYHMQZRENCY
|
7.0 | Ki | 29 | — | |
NSDIHUXUFJHXRA
|
7.0 | Ki | 11 | — | |
PBTNYNHOVGFGNO
|
7.0 | IC50 | 2 | — | |
TVUWQDLBEOZVOU
|
7.0 | IC50 | 41 | — | |
ZDPGLLQANLROFM
|
7.0 | Ki | 17 | — | |
ZYTFPHRVOZXPGZ
|
7.0 | Ki | 30 | — | |
PKOGEJUUQGCYAK
|
7.0 | IC50 | 3 | — | |
ZLNVBIGZYRPQKY
|
7.0 | IC50 | 15 | — | |
HLUQDCJXKVVBRH
|
7.0 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
7.0 | Kd | 29 | — | |
BKLVJGBLXVWFCJ
|
7.0 | IC50 | 3 | Yes | |
CIDXXRSLUUUBDG
|
7.0 | IC50 | 2 | — | |
FHDFIUFWMGMGTR
|
7.0 | IC50 | 5 | — | |
JOKSIWLEZWYCLI
|
7.0 | IC50 | 2 | — | |
XOXWOPNBJDVSJP
|
7.0 | Ki | 8 | — | |
ZSSHCAVAAPDLII
|
7.0 | IC50 | 5 | — | |
JYRJOQGKGMHTOO
|
7.0 | IC50 | 11 | — | |
SVZINFYUFRYAEN
|
7.0 | IC50 | 2 | — |