Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJXVAAHYUFZELV
|
8.3 | IC50 | 6 | — | |
SSIOYGMEKCPFAV
|
8.3 | IC50 | 5 | — | |
YNRGKDBIZBNELI
|
8.3 | IC50 | 3 | — | |
JNWDMRNNBZSXQY
|
8.3 | IC50 | 2 | — | |
LERGEXSFRXRSFX
|
8.3 | Ki | 4 | — | |
SJWPQHGIWPYOHJ
|
8.3 | IC50 | 2 | — | |
XZRIWFSNYJOZDQ
|
8.3 | Ki | 4 | — | |
YERVFCNDCWMBBO
|
8.3 | IC50 | 3 | — | |
YFRIHUMUDOXHTG
|
8.3 | IC50 | 5 | — | |
ZYONZFOMVOBYKS
|
8.3 | IC50 | 3 | — | |
BNHMMYCGPSNDMA
|
8.3 | Ki | 4 | — | |
FTPNAFTXRYWIHM
|
8.3 | Ki | 4 | — | |
KHUHONPSWMPDIC
|
8.3 | Ki | 4 | — | |
KHUHONPSWMPDIC
|
8.3 | Ki | 4 | — | |
QYGQOWFBQPSYJM
|
8.3 | Ki | 4 | — | |
UVVGSZJKQAELIC
|
8.3 | IC50 | 4 | — | |
YPJRHEKCFKOVRT
|
8.3 | IC50 | 12 | — | |
AVKHUGZDSUKIKQ
|
8.3 | IC50 | 3 | — | |
BENAWDZPBLPFCU
|
8.3 | IC50 | 3 | — | |
CFZGMAQTSTWGSI
|
8.3 | IC50 | 2 | — | |
GZVZVBKIIIOOOF
|
8.3 | Ki | 4 | — | |
GZVZVBKIIIOOOF
|
8.3 | Ki | 4 | — | |
KYMNNSMBWCZWCF
|
8.3 | IC50 | 6 | — | |
MLLWORSXSDVTQA
|
8.3 | IC50 | 2 | — | |
PDGKHKMBHVFCMG
|
8.3 | IC50 | 5 | — | |
PRGZEWRXEYVMGW
|
8.3 | Ki | 4 | — | |
XKPGLBSDWLZQRX
|
8.3 | IC50 | 2 | — | |
XXBMNYHUMYIUIC
|
8.3 | IC50 | 3 | — | |
YYWWXDBYEUYMKM
|
8.3 | IC50 | 3 | — | |
AWSGLYKKQMTOCZ
|
8.3 | IC50 | 3 | — | |
CXOZYBPVDKRPHI
|
8.3 | IC50 | 2 | — | |
HTIZPPSACKEUKK
|
8.3 | Ki | 4 | — | |
IIHKFIWSMAISST
|
8.3 | IC50 | 3 | — | |
LKPSCTJYYAVIIL
|
8.3 | IC50 | 3 | — | |
LMABWMJUORCNEW
|
8.3 | Ki | 4 | — | |
OJJODPGVVWMKKM
|
8.3 | Ki | 4 | — | |
OXTMSCZUAJMZIC
|
8.3 | IC50 | 2 | — | |
PFXDTPBJPRFRRN
|
8.3 | Ki | 4 | — | |
PLHTXTDCAFCNQE
|
8.3 | Ki | 4 | — | |
UHCMUGYUWQCODZ
|
8.3 | Ki | 4 | — | |
BAOXEYLXBCETRN
|
8.3 | Ki | 4 | — | |
CPJXTPZMRAOYPN
|
8.3 | IC50 | 2 | — | |
CZQMPFCNIINMMC
|
8.3 | IC50 | 8 | — | |
DYYOXQSHYDLEFT
|
8.3 | IC50 | 2 | — | |
DZKMAWNYSJECKX
|
8.3 | IC50 | 12 | — | |
IEPWMLWPYJPPOJ
|
8.3 | IC50 | 3 | — | |
IHNQNVXNYQNXFW
|
8.3 | IC50 | 3 | — | |
INUMHURQTSNMFM
|
8.3 | IC50 | 8 | — | |
LEKYSYXNVDOBCA
|
8.3 | IC50 | 5 | — | |
MRPVMOCAEFVNTQ
|
8.3 | IC50 | 3 | — |