Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FTPNAFTXRYWIHM
|
8.4 | Ki | 4 | — | |
KXFIUSMEECFBBN
|
8.4 | Ki | 6 | — | |
QPUBZAAAHLUCJC
|
8.4 | Ki | 4 | — | |
SKRUYIPFBIYOHZ
|
8.4 | IC50 | 2 | — | |
UZUCFTPPULEGQO
|
8.4 | IC50 | 9 | — | |
COWPKYBSZGEQGW
|
8.4 | Ki | 4 | — | |
MYKPWRUVZULGRH
|
8.4 | IC50 | 4 | — | |
UCTSPGHNUJSBEO
|
8.4 | IC50 | 2 | — | |
WTKYHVUVQSLNBW
|
8.4 | IC50 | 6 | — | |
ZAJRLIWINRGNKY
|
8.4 | IC50 | 6 | — | |
ZTXZICVBZWFLGQ
|
8.4 | IC50 | 3 | — | |
HZORGXNHDYOIAL
|
8.4 | IC50 | 3 | — | |
ICBZKFXPIBGECC
|
8.4 | IC50 | 3 | — | |
JRNJNYBQQYBCLE
|
8.4 | IC50 | 40 | Yes | |
MHBAURANSRCGRJ
|
8.4 | IC50 | 2 | — | |
PJAZUKUXPBWWHG
|
8.4 | IC50 | 2 | — | |
PJROIFLISSJQQQ
|
8.4 | IC50 | 4 | — | |
PSWOMNFIVDHMDM
|
8.4 | IC50 | 6 | — | |
RFEGHSBZJMLRST
|
8.4 | IC50 | 5 | — | |
RNHRCKQJHFBOKM
|
8.4 | IC50 | 2 | — | |
SLHUOQIIOYHUFR
|
8.4 | IC50 | 2 | — | |
VADHWSWHRRXKCV
|
8.4 | IC50 | 2 | — | |
XCTNQHXXOHMINL
|
8.4 | IC50 | 3 | — | |
XQCKNNHFNQYTHZ
|
8.4 | IC50 | 3 | — | |
XTSFMAFWRLGELC
|
8.4 | IC50 | 6 | — | |
YEQZZLYGLQFEAM
|
8.4 | IC50 | 3 | — | |
YUQBNHAASVYJAM
|
8.4 | IC50 | 2 | — | |
IPHOLKTXQVULGA
|
8.4 | IC50 | 9 | — | |
NPLHHQHEODJUBY
|
8.4 | IC50 | 6 | — | |
FGFWZFYILZKNBW
|
8.4 | IC50 | 6 | — | |
KMHNZVWSMBCPMT
|
8.4 | IC50 | 8 | — | |
KZZDDXBCJROTIP
|
8.4 | IC50 | 8 | — | |
MSKGFMBSNBBHMB
|
8.4 | IC50 | 2 | — | |
OCVMTGAKDLXKAY
|
8.4 | Ki | 4 | — | |
SSVSKCKWUAPYHI
|
8.4 | IC50 | 8 | — | |
UXLWEYWOVBRHJH
|
8.4 | Ki | 4 | — | |
ZGBMIKQTQVROES
|
8.4 | Ki | 4 | — | |
ZYOVPUHJYUVVBM
|
8.4 | Ki | 4 | — | |
JGNMMLNIOWYNHJ
|
8.4 | IC50 | 8 | — | |
QVISYMCZJFEAKJ
|
8.4 | Ki | 5 | — | |
YKDDWNDRNJMVDF
|
8.4 | IC50 | 4 | — | |
BYHCVEJLZXEHHO
|
8.4 | IC50 | 3 | — | |
KSCSDVHAZVSGAW
|
8.4 | Ki | 4 | — | |
MCPPMOSBWNMSOA
|
8.4 | IC50 | 5 | — | |
RKILQDBEPHSTGP
|
8.4 | IC50 | 4 | — | |
SOHOEERULHWXJB
|
8.4 | IC50 | 5 | — | |
TWTKMJWAXOPXSX
|
8.4 | IC50 | 5 | — | |
UXLWEYWOVBRHJH
|
8.4 | Ki | 4 | — | |
IIHKFIWSMAISST
|
8.3 | IC50 | 6 | — | |
JRHOBEGXOYAOBM
|
8.3 | Ki | 4 | — |