Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VGQBMNJRVGPBKT
|
8.5 | IC50 | 3 | — | |
ZFNZZKVYLDBWRD
|
8.5 | Ki | 8 | — | |
DLOAOZHQATYZNK
|
8.5 | IC50 | 2 | — | |
HOKDQPMWTBQYHL
|
8.5 | IC50 | 8 | — | |
XGQSZIVZWJHPHL
|
8.5 | IC50 | 2 | — | |
ZURIPGCQHWFPSQ
|
8.5 | IC50 | 2 | — | |
AYCUZAAKVCOJJW
|
8.5 | Ki | 4 | — | |
DSMBDRWDECFDNR
|
8.5 | IC50 | 7 | — | |
GKQHGPBOEGPFCT
|
8.5 | Ki | 4 | — | |
HWUQUQZRNDZMLC
|
8.5 | IC50 | 3 | — | |
YPMOBRWHNOTUIL
|
8.5 | IC50 | 7 | — | |
ZBYFYISKUULBLB
|
8.5 | Ki | 4 | — | |
ANELMUPUYRZVHZ
|
8.5 | IC50 | 7 | — | |
IDNJKMAZNUUVIO
|
8.5 | IC50 | 9 | — | |
JRGMQQCQWFMKLA
|
8.5 | IC50 | 6 | — | |
PACLAQXDVXULPW
|
8.5 | Ki | 4 | — | |
HWUQUQZRNDZMLC
|
8.5 | IC50 | 3 | — | |
IYLQAMPBXDBIFL
|
8.5 | IC50 | 2 | — | |
JSCXSRGTJHDPTA
|
8.5 | Ki | 4 | — | |
UDVJBRYBBSVDDS
|
8.5 | IC50 | 14 | — | |
XJKTXWSMMWPNTP
|
8.5 | IC50 | 6 | — | |
DECHPPWNVHMSRM
|
8.5 | Ki | 4 | — | |
JKKUZTDMJDZHEB
|
8.5 | IC50 | 7 | — | |
QHCHMOFMVBOPSK
|
8.5 | IC50 | 3 | — | |
SLORTXJSOVPUPP
|
8.5 | IC50 | 3 | — | |
XLZHLULRODUOPS
|
8.5 | IC50 | 5 | — | |
ZUOVZWHQGAJGQA
|
8.5 | IC50 | 3 | — | |
BLBRCCGITKEOBW
|
8.5 | IC50 | 3 | — | |
DSNHCXNKKZEERJ
|
8.5 | IC50 | 2 | — | |
DYNVDYWVVYCHHR
|
8.5 | IC50 | 3 | — | |
FEBXDTFBHZJUJT
|
8.5 | IC50 | 5 | — | |
FFNUKKIYDLQPQE
|
8.5 | Ki | 4 | — | |
FHEQFUUMLHFZOS
|
8.5 | IC50 | 3 | — | |
HCAPKVUYVLOOHA
|
8.5 | IC50 | 3 | — | |
JAMUFNNBMXMUIC
|
8.5 | IC50 | 3 | — | |
PFGMZHAOYLGYMA
|
8.5 | Ki | 4 | — | |
RFWCLSISMUZKNC
|
8.5 | Ki | 4 | — | |
UGMXVKWXOFIULK
|
8.5 | IC50 | 5 | — | |
ISWNVTVWJJQFQV
|
8.4 | IC50 | 3 | — | |
JDVCOPUEQIAVNW
|
8.4 | IC50 | 3 | — | |
LGDFLYMYRBSZOR
|
8.4 | Ki | 4 | — | |
NUGRJQBHFHUEGX
|
8.4 | Ki | 4 | — | |
MZGANASDMYZAGW
|
8.4 | IC50 | 3 | — | |
SRIUCPFRQBBONO
|
8.4 | Ki | 4 | — | |
VNRANBWAFHAFQG
|
8.4 | IC50 | 2 | — | |
WIAMCDYCLOMHKF
|
8.4 | IC50 | 6 | — | |
DHPLYCJQWJHXFH
|
8.4 | IC50 | 3 | — | |
GEZUTMXESRSXNV
|
8.4 | Ki | 4 | — | |
QXBRBWDRQIISAT
|
8.4 | IC50 | 6 | — | |
BTTJTCLIZBSDNP
|
8.4 | IC50 | 8 | — |