Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBYFYISKUULBLB
|
8.6 | Ki | 4 | — | |
ANDYPXVQXOKMKT
|
8.6 | IC50 | 3 | — | |
ROVFHHODJNANCC
|
8.6 | IC50 | 2 | — | |
UKVZKVRVVNTCMR
|
8.6 | Ki | 4 | — | |
WIAMCDYCLOMHKF
|
8.6 | IC50 | 3 | — | |
CVNQRFZZFGTWIK
|
8.6 | IC50 | 3 | — | |
DHROAMIZLTYJCT
|
8.6 | Ki | 4 | — | |
DSUXSBZUWGKTQG
|
8.6 | IC50 | 2 | — | |
IVKYJVDFJKEXIH
|
8.6 | IC50 | 6 | — | |
SDAWBLGFXWXOCC
|
8.6 | IC50 | 3 | — | |
TWNUIDQVTSUXKY
|
8.6 | IC50 | 3 | — | |
UPAMTEZWUWUYNR
|
8.6 | IC50 | 2 | — | |
ZJXAYHKSLDKUOY
|
8.6 | IC50 | 3 | — | |
ZQHZICOJSNIGEO
|
8.6 | IC50 | 2 | — | |
FIFYTWABWYHZIS
|
8.6 | Ki | 4 | — | |
GZAGBRPFBCDRDL
|
8.6 | IC50 | 4 | — | |
JINXSJRUNKRAKJ
|
8.6 | IC50 | 3 | — | |
LCDCVRYMEWMBEV
|
8.6 | IC50 | 5 | — | |
MDQNQFYRPHYQNJ
|
8.6 | Ki | 4 | — | |
QXZISVGKZJBIFK
|
8.6 | IC50 | 2 | — | |
SUEYATVNHWMTSO
|
8.6 | IC50 | 7 | — | |
WQGCPJJNZKLUAU
|
8.6 | IC50 | 4 | — | |
SSIDJRGNBKXDGV
|
8.6 | IC50 | 8 | — | |
XZKHOZLKTBKGNZ
|
8.6 | Ki | 4 | — | |
GFUYDGPHKDLMHQ
|
8.6 | IC50 | 2 | — | |
LQLWCEYRAKKEIP
|
8.6 | IC50 | 2 | — | |
PPBUGSNWRZPWMZ
|
8.6 | Ki | 4 | — | |
RKUPKTQQPJAABW
|
8.6 | Ki | 2 | — | |
SALMKXDVOXFTFG
|
8.6 | IC50 | 3 | — | |
WFMBBNNZNAMTGD
|
8.6 | Ki | 7 | — | |
XFCBYRQZMFSMHZ
|
8.6 | Ki | 4 | — | |
DCRIEDZZYPOGPK
|
8.5 | IC50 | 4 | — | |
DVAPMYJVUZJNDK
|
8.5 | Ki | 8 | — | |
GNEARXSVRDSWKT
|
8.5 | IC50 | 7 | — | |
UQNXGQYESHUBBX
|
8.5 | IC50 | 3 | — | |
UTDIUAOBXDHROL
|
8.5 | IC50 | 5 | — | |
WJENEGQQOQWXTQ
|
8.5 | IC50 | 3 | — | |
LIJUCWLALFXGCL
|
8.5 | IC50 | 7 | — | |
AYTDCXHHGYDWLU
|
8.5 | IC50 | 3 | — | |
CGZPQEKNAAVWHA
|
8.5 | Ki | 4 | — | |
HMUKVTQDAZQBHU
|
8.5 | IC50 | 2 | — | |
JYLSDMOABXIYSW
|
8.5 | IC50 | 3 | — | |
KZTHERIRWPUOBR
|
8.5 | Ki | 4 | — | |
LUHGNQLUGTWNCL
|
8.5 | Ki | 12 | — | |
LXWKFZODCMNRLB
|
8.5 | IC50 | 3 | — | |
MGOBPQYJSRWRLP
|
8.5 | IC50 | 3 | — | |
QFGDMFUYBQHULK
|
8.5 | IC50 | 3 | — | |
RLWUWLYKPWQOFL
|
8.5 | IC50 | 3 | — | |
SESXHBRHIPVWPS
|
8.5 | IC50 | 3 | — | |
UFUZVHSCAUVFOR
|
8.5 | IC50 | 5 | — |