Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QSPGRGDMJHWLAB
|
6.2 | IC50 | 2 | — | |
UCZKCMDYRWWWAW
|
6.2 | IC50 | 2 | — | |
AMPVAHRRWJJJOA
|
6.2 | IC50 | 2 | — | |
AWUZKGRBVIKLQF
|
6.2 | IC50 | 2 | — | |
BNFWUGLGTHBKHE
|
6.2 | IC50 | 2 | — | |
CHUDIJJINHPGKN
|
6.2 | IC50 | 6 | — | |
JXDLWPHADRZUDZ
|
6.2 | IC50 | 2 | — | |
ATBAETXFFCOZOY
|
6.2 | IC50 | 39 | — | |
ATMUPWYSEDBDPX
|
6.2 | IC50 | 2 | — | |
KPSNDCVFVSQFFH
|
6.2 | IC50 | 2 | — | |
ASDDTGMTDPGXHC
|
6.2 | IC50 | 2 | — | |
BXQKMGAINGBZAW
|
6.2 | IC50 | 11 | — | |
HBNWVIQVJCNKNS
|
6.2 | IC50 | 2 | — | |
PBJCSRINGCPRJY
|
6.2 | IC50 | 2 | — | |
GRHFKIYSAMODSD
|
6.1 | Ki | 7 | — | |
CBIGSGRHQIOPQH
|
6.1 | IC50 | 2 | — | |
RUCZHYZBUIFIFW
|
6.1 | IC50 | 2 | — | |
UNGSBCKKKYIIJC
|
6.1 | IC50 | 6 | Yes | |
ZAZNEIMFYPXDMS
|
6.1 | IC50 | 4 | — | |
ZWZDGQSAMQVAHB
|
6.1 | IC50 | 2 | — | |
AJXAXQOBZWUUQX
|
6.1 | IC50 | 2 | — | |
CHMCDQVKNOFOSV
|
6.1 | IC50 | 2 | — | |
WIXACQKVOOJSHW
|
6.1 | IC50 | 2 | — | |
WIZPFVWZYLEGII
|
6.1 | IC50 | 6 | — | |
ZFVBEQZSPYFLJB
|
6.1 | IC50 | 5 | — | |
AWUZKGRBVIKLQF
|
6.1 | IC50 | 2 | — | |
GWGVHVMHVZRQJD
|
6.1 | IC50 | 2 | — | |
KFALTJHKAYBGIC
|
6.1 | IC50 | 2 | — | |
MPNFAZGZWVPCCV
|
6.1 | IC50 | 2 | — | |
QFWSAIKNLPPPHT
|
6.1 | IC50 | 2 | — | |
DMCIVYAQQSYXTQ
|
6.1 | IC50 | 2 | — | |
QRPJDQZOXSLSEK
|
6.1 | IC50 | 11 | — | |
SNSZKJPBYIHUPY
|
6.1 | IC50 | 2 | — | |
CLCKDDAPJRHFEN
|
6.1 | IC50 | 9 | — | |
GYKQZNKJVUESID
|
6.1 | IC50 | 2 | — | |
KNSQRKGMNUEWEC
|
6.1 | IC50 | 2 | — | |
TWQNXXRFGMYDMQ
|
6.1 | IC50 | 5 | — | |
UZQXPHDZFUAMQS
|
6.1 | IC50 | 9 | — | |
VLDDBBJMBQBNEJ
|
6.1 | IC50 | 2 | — | |
DMCIVYAQQSYXTQ
|
6.1 | IC50 | 2 | — | |
FFNPBRFKICWUCS
|
6.1 | IC50 | 2 | — | |
HKTDZTIJYNTRCQ
|
6.1 | IC50 | 2 | — | |
ANQYGTSNOCQORM
|
6.1 | IC50 | 2 | — | |
FWKJOFFEPRZHEJ
|
6.1 | IC50 | 2 | — | |
VSWIXDIHGDTNBN
|
6.1 | IC50 | 2 | — | |
BAJWJQKHEVLEIH
|
6.0 | IC50 | 5 | — | |
CYQVUZINNHQLBF
|
6.0 | IC50 | 2 | — | |
GGZVKRXAOUQBQV
|
6.0 | IC50 | 5 | — | |
WOELEDNHQCSWNR
|
6.0 | IC50 | 3 | — | |
DIRJXVHFPSKLII
|
6.0 | IC50 | 2 | — |