Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YLOQURWWSGPVHD
|
6.3 | IC50 | 2 | — | |
YQVYMELPOPTNDV
|
6.3 | IC50 | 3 | — | |
YTRZTOPIENEURB
|
6.3 | IC50 | 5 | — | |
YUOHLMLGTIBJMB
|
6.3 | IC50 | 4 | — | |
YWLAOJSVGLKWDA
|
6.3 | IC50 | 3 | — | |
YXQIJCZYWYSLMZ
|
6.3 | IC50 | 4 | — | |
ZBKDFCCYRATMJF
|
6.3 | IC50 | 3 | — | |
ZWKJWQSYJYMAPM
|
6.3 | IC50 | 2 | — | |
ZYIUATVXCNVESH
|
6.3 | IC50 | 6 | — | |
BGLKUMXXQFFELV
|
6.2 | IC50 | 2 | — | |
BRSLFMLGEMXLEU
|
6.2 | IC50 | 2 | — | |
FHIVDVRFOQWJJD
|
6.2 | IC50 | 2 | — | |
LGOXNTCIROJSQM
|
6.2 | IC50 | 2 | — | |
FCKWPUFNPAWKRB
|
6.2 | IC50 | 2 | — | |
HVWJXUQLUOVWFM
|
6.2 | IC50 | 3 | — | |
LKTWMXPIHJGMOH
|
6.2 | IC50 | 2 | — | |
QAKQOZHFKOCBPL
|
6.2 | IC50 | 2 | — | |
UCSSXRJZMVWANS
|
6.2 | IC50 | 2 | — | |
YPSCKJWJIXZMSC
|
6.2 | IC50 | 15 | — | |
AESLLIYWIJHRIE
|
6.2 | IC50 | 2 | — | |
CKZXLBVKAYSONS
|
6.2 | IC50 | 5 | — | |
DQKKUVSYKRLEBM
|
6.2 | IC50 | 10 | — | |
KAVSBZSFIXQLLS
|
6.2 | IC50 | 2 | — | |
PAJDGKAXRPLQSA
|
6.2 | IC50 | 2 | — | |
PHYKSMUMABKXEB
|
6.2 | IC50 | 2 | — | |
PQAJMNITAQGSCS
|
6.2 | IC50 | 9 | — | |
ABXJEHDBGMUMPY
|
6.2 | IC50 | 2 | — | |
DGPVLDATMHPRMS
|
6.2 | IC50 | 2 | — | |
DZIDIUZYNSZKTB
|
6.2 | IC50 | 2 | — | |
HLCKDKMRGSCDRW
|
6.2 | IC50 | 5 | — | |
JJKRSPZQJWOKSJ
|
6.2 | IC50 | 2 | — | |
KZNAEWYKSFFELV
|
6.2 | IC50 | 2 | — | |
QSPGRGDMJHWLAB
|
6.2 | IC50 | 2 | — | |
USSLYTCUOBWSFG
|
6.2 | IC50 | 3 | — | |
LPKPAAYYOJMPCW
|
6.2 | IC50 | 2 | — | |
MPNFAZGZWVPCCV
|
6.2 | IC50 | 2 | — | |
OFGFMPRVIBGFKB
|
6.2 | IC50 | 2 | — | |
BNFWUGLGTHBKHE
|
6.2 | IC50 | 2 | — | |
ZDEBEWQYXJZQRS
|
6.2 | IC50 | 12 | — | |
HSRVWDOXTFEAGX
|
6.2 | IC50 | 2 | — | |
LPGAZCZIRANIGC
|
6.2 | IC50 | 2 | — | |
MDZBKUVFDTVNSE
|
6.2 | IC50 | 2 | — | |
MXTOHVOXLMRCLK
|
6.2 | IC50 | 2 | — | |
TVZKWMUWNDZPCZ
|
6.2 | IC50 | 2 | — | |
UYIAGEDEEBGQRM
|
6.2 | IC50 | 2 | — | |
YUFVQEHKXVADND
|
6.2 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.2 | IC50 | 12 | Yes | |
LPKPAAYYOJMPCW
|
6.2 | IC50 | 2 | — | |
MIJGGHANRDZXTD
|
6.2 | IC50 | 3 | — | |
MXPOUDOWVQWPSA
|
6.2 | IC50 | 2 | — |