Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DEUZACBXMBZZRF
|
6.3 | Ki | 4 | — | |
FYDJUDIQVFDSPD
|
6.3 | IC50 | 2 | — | |
JTIFUJUJDWUQEV
|
6.3 | IC50 | 12 | — | |
SKBWHULYERLNLR
|
6.3 | IC50 | 2 | — | |
ARZCNFVGTWMROY
|
6.3 | IC50 | 6 | — | |
AXRXMZKVXARJEN
|
6.3 | IC50 | 3 | — | |
BFTPBRJJWBLTEE
|
6.3 | IC50 | 5 | — | |
BHEVXPKVRPTJTA
|
6.3 | IC50 | 5 | — | |
BIWBSWKCOJWZND
|
6.3 | IC50 | 2 | — | |
BKLHNPDHXKQVRD
|
6.3 | IC50 | 2 | — | |
CFJROUOQZZNEHG
|
6.3 | IC50 | 3 | — | |
CNPCDJLCMSGEOJ
|
6.3 | IC50 | 2 | — | |
CPPKSKHDVMJSGS
|
6.3 | IC50 | 4 | — | |
CPPKSKHDVMJSGS
|
6.3 | IC50 | 3 | — | |
CXABQNFLIBANJT
|
6.3 | IC50 | 3 | — | |
DCIHHIYPTRKGLA
|
6.3 | IC50 | 3 | — | |
DIVSTSBKLAEJDM
|
6.3 | IC50 | 2 | — | |
DJBDVEQBCUISBP
|
6.3 | IC50 | 2 | — | |
DODICJSQANDMOW
|
6.3 | IC50 | 3 | — | |
DUAHUWZSSCBNCQ
|
6.3 | IC50 | 5 | — | |
FEJHIDUOCKGDJQ
|
6.3 | IC50 | 2 | — | |
FHRXQRGKKCMVHS
|
6.3 | IC50 | 2 | — | |
GPSDEPYWJYUQER
|
6.3 | IC50 | 2 | — | |
GQKLNZLOCNSFOD
|
6.3 | IC50 | 2 | — | |
GSTJDNPGSVZHDA
|
6.3 | IC50 | 2 | — | |
HCBVVIFOIUAUCN
|
6.3 | IC50 | 3 | — | |
HOISFQJJCQCQFV
|
6.3 | IC50 | 5 | — | |
HRXOXTKKMBFOQP
|
6.3 | IC50 | 3 | — | |
IGLHISZMQZPVOP
|
6.3 | IC50 | 4 | — | |
IGLHISZMQZPVOP
|
6.3 | IC50 | 3 | — | |
JDUIELGVEPIVMG
|
6.3 | IC50 | 4 | — | |
JXASPAXWKIGRSO
|
6.3 | IC50 | 2 | — | |
KDQKJDYKGJRHRE
|
6.3 | IC50 | 3 | — | |
KQXQWLRLPZKNES
|
6.3 | IC50 | 2 | — | |
KTYZEMCWKVWKOX
|
6.3 | IC50 | 2 | — | |
KXDROPRNEYFQHH
|
6.3 | IC50 | 5 | — | |
LYXRABIWUDHHOT
|
6.3 | IC50 | 4 | — | |
MAWZHASBBDEYSI
|
6.3 | IC50 | 2 | — | |
MCVYLHWRTAZNNE
|
6.3 | IC50 | 6 | — | |
MVBOUBNVEXSMFL
|
6.3 | IC50 | 2 | — | |
MWILTCFDLRXJDY
|
6.3 | IC50 | 4 | — | |
NBOMRDUNYYSFKM
|
6.3 | IC50 | 4 | — | |
NHURAJZSHKFCNL
|
6.3 | IC50 | 5 | — | |
NYNILZXULKMIKC
|
6.3 | IC50 | 2 | — | |
OBLJLYMRPRWYFS
|
6.3 | IC50 | 2 | — | |
OELWRYRKFMYGJW
|
6.3 | IC50 | 4 | — | |
OQEZTXDNCMJLDJ
|
6.3 | IC50 | 3 | — | |
OURKCQIQALLKJV
|
6.3 | IC50 | 3 | — | |
OVQMEODZAKFJGT
|
6.3 | IC50 | 2 | — | |
OWNAKRKOXLNXIK
|
6.3 | IC50 | 2 | — |