Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUTNEOKLYIUETI
|
6.4 | IC50 | 2 | — | |
ZZABWRAOQNGARP
|
6.4 | IC50 | 2 | — | |
GDDLWKLTUNDNCJ
|
6.4 | IC50 | 2 | — | |
NUBBIJVOSXWZTF
|
6.4 | IC50 | 13 | — | |
QBTKCYHFYXSRAI
|
6.4 | IC50 | 2 | — | |
CEBMEQPREMCWOL
|
6.4 | IC50 | 7 | — | |
GKQOHITZTWZGRC
|
6.4 | IC50 | 2 | — | |
QAKQOZHFKOCBPL
|
6.4 | IC50 | 2 | — | |
GMUOLFXLMDSJBA
|
6.4 | IC50 | 2 | — | |
TUICYWDMLMCHGT
|
6.4 | IC50 | 2 | — | |
YAGLZRLKRDTHPW
|
6.4 | IC50 | 4 | — | |
JRRRQHJGIOSHEE
|
6.3 | IC50 | 2 | — | |
LOYSCNBYDPTSAA
|
6.3 | Ki | 10 | — | |
NPQSOFKMVBBVFF
|
6.3 | IC50 | 2 | — | |
QOEIEBLLVFISRF
|
6.3 | IC50 | 2 | — | |
SLLDMBDDRHKGKF
|
6.3 | IC50 | 2 | — | |
YLKRCKNIKRAUQP
|
6.3 | IC50 | 2 | — | |
BZWJJBNGNGVBMX
|
6.3 | IC50 | 4 | — | |
WMHURJYFLDPMEB
|
6.3 | IC50 | 6 | — | |
XCCCFEGJPRCHRL
|
6.3 | IC50 | 7 | — | |
BXPPINFBXDOAPI
|
6.3 | IC50 | 2 | — | |
MDZBKUVFDTVNSE
|
6.3 | IC50 | 2 | — | |
MPYGRCKAAVICEA
|
6.3 | IC50 | 5 | — | |
MTNBRBDFNSGQKB
|
6.3 | Ki | 10 | — | |
OCQGVQNZFLPPRL
|
6.3 | IC50 | 2 | — | |
VEFPYYIJHHBRQO
|
6.3 | IC50 | 2 | — | |
CBIGSGRHQIOPQH
|
6.3 | IC50 | 2 | — | |
HBNWVIQVJCNKNS
|
6.3 | IC50 | 2 | — | |
LQHROIHZWLXWTM
|
6.3 | IC50 | 2 | — | |
MOXBYMQBYZTOJA
|
6.3 | IC50 | 11 | — | |
NZTXMMVRWPITFU
|
6.3 | IC50 | 2 | — | |
TVZKWMUWNDZPCZ
|
6.3 | IC50 | 2 | — | |
TVZKWMUWNDZPCZ
|
6.3 | IC50 | 2 | — | |
ZLNVBIGZYRPQKY
|
6.3 | IC50 | 15 | — | |
QSPGRGDMJHWLAB
|
6.3 | IC50 | 2 | — | |
STIWJUXFYZIOEQ
|
6.3 | IC50 | 2 | — | |
XYWLVOJJDGXVRI
|
6.3 | IC50 | 2 | — | |
YTCPGIQPAHCLSI
|
6.3 | Ki | 4 | — | |
HGYGADURLZIPNZ
|
6.3 | IC50 | 2 | — | |
VPDSZVYUHWYXCW
|
6.3 | IC50 | 6 | — | |
WEHVSGDBAMEZCL
|
6.3 | IC50 | 2 | — | |
XJSSBCWQSJYAAR
|
6.3 | IC50 | 2 | — | |
DTYXXTKHTSQKFJ
|
6.3 | IC50 | 2 | — | |
GAVPKFXPGFHFSY
|
6.3 | IC50 | 7 | Yes | |
QAJVTVKGYCSHLP
|
6.3 | IC50 | 2 | — | |
NLKSAJZXMQSXKO
|
6.3 | IC50 | 2 | — | |
ODDUUXAHBDCKIJ
|
6.3 | IC50 | 11 | — | |
PXHMGBDEPBEGQH
|
6.3 | IC50 | 2 | — | |
ZCZWCPYCSYTXDF
|
6.3 | IC50 | 2 | — | |
AYTLDMIYGVIYLM
|
6.3 | IC50 | 2 | — |