Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JPYDPHLKOMGSJO
|
6.5 | IC50 | 2 | — | |
KGJVKYSVVOQPDL
|
6.5 | IC50 | 13 | — | |
KGPWFLJNWXSMCR
|
6.5 | IC50 | 2 | — | |
NNPRQBLRXNNMJV
|
6.5 | IC50 | 5 | — | |
NUEFFTPUFYWSFG
|
6.5 | IC50 | 2 | — | |
PFALOULACVHTOP
|
6.5 | IC50 | 2 | — | |
PZVOIGICALCYSF
|
6.5 | IC50 | 3 | — | |
QTBZFGYORPEJEV
|
6.5 | IC50 | 3 | — | |
SNPPXRDRBRHKMN
|
6.5 | IC50 | 3 | — | |
TYFRBVNZVSBSKA
|
6.5 | IC50 | 2 | — | |
UZLSPPARRYQODK
|
6.5 | IC50 | 2 | — | |
WZBGAJOCGTZFCV
|
6.5 | IC50 | 3 | — | |
XRYOBKDKPBPRIT
|
6.5 | IC50 | 3 | — | |
XVGRWDWWYUTWLD
|
6.5 | IC50 | 2 | — | |
ZTSRCWHLXVMIPQ
|
6.5 | IC50 | 3 | — | |
AAYPLLWGPJQWCC
|
6.5 | IC50 | 15 | Yes | |
DVULGARGBYQBPJ
|
6.5 | IC50 | 2 | — | |
TYWICOYJWWRAAG
|
6.5 | IC50 | 2 | — | |
VDSHZLHHBAROJU
|
6.5 | IC50 | 2 | — | |
ZNAVDFQDONRFBI
|
6.5 | IC50 | 2 | — | |
AVIWDYSJSPOOAR
|
6.4 | IC50 | 11 | — | |
BZXZKWSLTSIOMY
|
6.4 | IC50 | 2 | — | |
DGPVLDATMHPRMS
|
6.4 | IC50 | 2 | — | |
NMEQPNSVTTWBOJ
|
6.4 | IC50 | 2 | — | |
ULAJBCKHKLTBJU
|
6.4 | IC50 | 2 | — | |
ZQJBROQJONVIEC
|
6.4 | IC50 | 2 | — | |
ATMUPWYSEDBDPX
|
6.4 | IC50 | 2 | — | |
CZMFKHZKGYYFSP
|
6.4 | IC50 | 3 | — | |
GYFQTLMDYXNZPR
|
6.4 | IC50 | 2 | — | |
NSJFZIYYYKMTMJ
|
6.4 | IC50 | 2 | — | |
QMFQNXRGLSNRKW
|
6.4 | IC50 | 2 | — | |
LVKJKRHVKKFITG
|
6.4 | IC50 | 2 | — | |
FIFUHCDTTSHUQT
|
6.4 | IC50 | 2 | — | |
FNAZUFVXFZSHAN
|
6.4 | IC50 | 3 | — | |
MTXGSPNFOOITQW
|
6.4 | IC50 | 2 | — | |
UYDMDSBIXKYMQD
|
6.4 | IC50 | 5 | — | |
VKGGKBNGOLFDMX
|
6.4 | IC50 | 2 | — | |
ZZBUMHLUAAJMOY
|
6.4 | IC50 | 2 | — | |
CMAOXPXXZOSIJY
|
6.4 | IC50 | 2 | — | |
HKLMPEVOJSPPJG
|
6.4 | IC50 | 2 | — | |
KDYHURHHRIDGQT
|
6.4 | IC50 | 4 | — | |
KOZFSFOOLUUIGY
|
6.4 | Kd | 88 | Yes | |
LXRJNNLNUWGVCX
|
6.4 | IC50 | 10 | — | |
QLUYMIVVAYRECT
|
6.4 | IC50 | 13 | — | |
URRIHRKEWFRNLT
|
6.4 | IC50 | 2 | — | |
WSGLUFHKWDKYLV
|
6.4 | IC50 | 2 | — | |
ZNAVDFQDONRFBI
|
6.4 | IC50 | 2 | — | |
NIXRABVGGAIGEC
|
6.4 | IC50 | 2 | — | |
NIXRABVGGAIGEC
|
6.4 | IC50 | 2 | — | |
OXFMTURCMJXJOI
|
6.4 | IC50 | 6 | — |