Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADCIWACTHXRXCW
|
6.6 | IC50 | 2 | — | |
BKIBIERXNSLGOL
|
6.6 | IC50 | 2 | — | |
DNURQZGRRIHXKJ
|
6.6 | IC50 | 2 | — | |
RRQMONAJNHHQCC
|
6.6 | IC50 | 2 | — | |
SKJMONQADFDYMK
|
6.6 | IC50 | 2 | — | |
VEBWDBXHNZZYSO
|
6.6 | IC50 | 2 | — | |
DADZAXRKSGGBOW
|
6.5 | IC50 | 2 | — | |
DCWNCWYHYUMEFR
|
6.5 | IC50 | 2 | — | |
NAGFLZVMWVHHLW
|
6.5 | Ki | 2 | — | |
RSQPNXBTPUXMQN
|
6.5 | IC50 | 12 | — | |
UKOWGHRRBISLOO
|
6.5 | IC50 | 2 | — | |
WHDHBZVTAJDTDO
|
6.5 | IC50 | 10 | — | |
ZPOSVRUJUALHAX
|
6.5 | IC50 | 2 | — | |
APOKZJTZDBUNNV
|
6.5 | IC50 | 4 | — | |
JFYAFMMSOVKSEU
|
6.5 | IC50 | 4 | — | |
NDLAFOKSJSLKGG
|
6.5 | IC50 | 4 | — | |
QECBYHQRTUOPOS
|
6.5 | IC50 | 2 | — | |
QECBYHQRTUOPOS
|
6.5 | IC50 | 2 | — | |
VJKHPOMKSRNBGY
|
6.5 | IC50 | 2 | — | |
GEFYRVKALMUFSB
|
6.5 | IC50 | 2 | — | |
IXLNTZGFRNXEDC
|
6.5 | IC50 | 3 | — | |
PPUUFIDXXJCITR
|
6.5 | IC50 | 4 | — | |
UPHNXAZSYZQUCI
|
6.5 | IC50 | 4 | — | |
VSHURSPEQITHNX
|
6.5 | IC50 | 4 | — | |
AGPQNNSQYCHUHR
|
6.5 | IC50 | 5 | — | |
BFSMGDJOXZAERB
|
6.5 | Kd | 33 | — | |
DZJCNUNAIXWMLJ
|
6.5 | IC50 | 2 | — | |
GLEPOVWXFFRWSW
|
6.5 | IC50 | 2 | — | |
NQRZZYMZECRALA
|
6.5 | IC50 | 2 | — | |
GKQOHITZTWZGRC
|
6.5 | IC50 | 2 | — | |
GUPLVXQEYAKBCK
|
6.5 | IC50 | 3 | — | |
ZMVQNBBXGBZQSY
|
6.5 | IC50 | 2 | — | |
AORLTNNDHWCLMA
|
6.5 | IC50 | 2 | — | |
CAWOMBHGPUUCGE
|
6.5 | IC50 | 4 | — | |
QRKQXCYYQSZGBN
|
6.5 | IC50 | 2 | — | |
GIAAALWHPIBJMG
|
6.5 | IC50 | 2 | — | |
PVCZVEAVKLUVDX
|
6.5 | IC50 | 2 | — | |
QECBYHQRTUOPOS
|
6.5 | IC50 | 2 | — | |
RDOKVGWGKMHBMG
|
6.5 | IC50 | 9 | — | |
UGRAFLUUHGUBAR
|
6.5 | IC50 | 2 | — | |
WFMZKYFCWOCGDW
|
6.5 | IC50 | 2 | — | |
AKAXSKGPOBYDLI
|
6.5 | IC50 | 2 | — | |
BYBKANFSSKDHSG
|
6.5 | IC50 | 2 | — | |
DDGUGNCWPAZRIR
|
6.5 | IC50 | 2 | — | |
DEXZHKNXZYDRKP
|
6.5 | IC50 | 2 | — | |
FPABGBDCJJVTMH
|
6.5 | IC50 | 3 | — | |
GBKKRKQHJUNMHL
|
6.5 | IC50 | 3 | — | |
HAGBYNGHDUURQD
|
6.5 | IC50 | 2 | — | |
IPJSMYHYHWQEMJ
|
6.5 | IC50 | 2 | — | |
JHKPHCUOXCKBCO
|
6.5 | IC50 | 2 | — |