Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNECPTZUDOQLHE
|
6.7 | IC50 | 2 | — | |
UNPMPNKARZANGA
|
6.7 | IC50 | 2 | — | |
WLTRIWCDHOZNRP
|
6.7 | IC50 | 14 | — | |
XKFYFHYPIPRAIB
|
6.7 | IC50 | 2 | — | |
ZJKDYTFNXUBLEQ
|
6.7 | IC50 | 15 | — | |
DEJMDEDQXYDMOK
|
6.7 | IC50 | 2 | — | |
FCLBVILBAPMKST
|
6.7 | IC50 | 13 | — | |
HWEBFAZCYKVEJD
|
6.7 | IC50 | 5 | — | |
VKZHSGOJYOUKNB
|
6.7 | Ki | 5 | — | |
HYDOSWLWKXMOGK
|
6.7 | IC50 | 2 | — | |
TVXXLAJWEQEGRC
|
6.7 | IC50 | 2 | — | |
MRERFRKMDQOLEP
|
6.7 | IC50 | 2 | — | |
PONGJVYMOPSJRY
|
6.7 | IC50 | 2 | — | |
XOHHDQPVPBYXEK
|
6.7 | IC50 | 2 | — | |
DEHFINBXRGBIHZ
|
6.6 | IC50 | 2 | — | |
HRKCERYJQXATNH
|
6.6 | IC50 | 11 | — | |
OBJNQQWSNUSMIU
|
6.6 | IC50 | 3 | — | |
PHZDWQYTFQOSSZ
|
6.6 | IC50 | 15 | — | |
UONTVBODKZAAKG
|
6.6 | IC50 | 6 | Yes | |
YENNZDUKQZAEML
|
6.6 | IC50 | 2 | — | |
CMJFZMMVFSMCTJ
|
6.6 | IC50 | 2 | — | |
OVLZNLFIVGBMBP
|
6.6 | IC50 | 2 | — | |
QXVWBJROURLRIW
|
6.6 | IC50 | 11 | — | |
PZBGPBZPHFHRHQ
|
6.6 | IC50 | 2 | — | |
VDSHZLHHBAROJU
|
6.6 | IC50 | 2 | — | |
FLXBKICISVDLQT
|
6.6 | IC50 | 2 | — | |
LUWQTRGZKXLDSO
|
6.6 | IC50 | 11 | — | |
MGENEBPUTRSHKN
|
6.6 | IC50 | 2 | — | |
BQMTVHKMQWOWGD
|
6.6 | IC50 | 2 | — | |
MBIXOXMOHXFUFZ
|
6.6 | IC50 | 3 | — | |
OVAITXNWYOTUTR
|
6.6 | IC50 | 2 | — | |
WDPQQGKAKPLXAJ
|
6.6 | IC50 | 4 | — | |
WIXACQKVOOJSHW
|
6.6 | IC50 | 2 | — | |
YBJLQBOUQXKRET
|
6.6 | Ki | 5 | — | |
YUOVFFUJYPBUGE
|
6.6 | IC50 | 2 | — | |
AKFBBBYLSSSRMT
|
6.6 | IC50 | 2 | — | |
BHWIQYBTLGGGBK
|
6.6 | IC50 | 2 | — | |
NASHAYHCDKSVRA
|
6.6 | Ki | 4 | — | |
OMBJFZLNXXKWTQ
|
6.6 | IC50 | 2 | — | |
OUSRERDVPWMEJK
|
6.6 | IC50 | 2 | — | |
QOTOLYJLZGPXEV
|
6.6 | IC50 | 2 | — | |
YITZLEHWDLDKBR
|
6.6 | IC50 | 2 | — | |
WFUYDZFIDJMSKL
|
6.6 | IC50 | 2 | — | |
HUNWQLBOLVYRMW
|
6.6 | IC50 | 11 | — | |
IYUGPEZCKNVRDO
|
6.6 | IC50 | 2 | — | |
MYSCCSFDIPYMDY
|
6.6 | IC50 | 3 | — | |
OBKJRYFTQJNTFG
|
6.6 | IC50 | 2 | — | |
OGSBFBXJSCWWMC
|
6.6 | IC50 | 2 | — | |
UXEWCQUEOJJYLF
|
6.6 | IC50 | 6 | — | |
WLPDYLPFPWPYBC
|
6.6 | IC50 | 11 | — |