Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMCUBSCEQXEGSP
|
6.8 | IC50 | 8 | — | |
VFCDEOOGPZZACO
|
6.8 | IC50 | 2 | — | |
DQMDXHWHDMGPCC
|
6.8 | IC50 | 6 | — | |
FILLLYJLVXSRAT
|
6.8 | IC50 | 4 | — | |
KSGRHPFFOUUFPR
|
6.8 | IC50 | 8 | — | |
MZKFILOLSANFFN
|
6.8 | IC50 | 8 | — | |
UELAYOOTACICFN
|
6.8 | IC50 | 2 | — | |
VUZDQQHRXMACQX
|
6.8 | IC50 | 2 | — | |
WPBMZKYEKGWUGB
|
6.8 | IC50 | 2 | — | |
YQOZFMRCEONJEU
|
6.8 | IC50 | 13 | — | |
FYDJUDIQVFDSPD
|
6.8 | IC50 | 2 | — | |
MSPUGHMWVNBVIW
|
6.8 | IC50 | 2 | — | |
NMXTWKFAOLSJAL
|
6.8 | IC50 | 3 | — | |
NZTXMMVRWPITFU
|
6.8 | IC50 | 2 | — | |
OVPNQJVDAFNBDN
|
6.8 | IC50 | 44 | Yes | |
STIWJUXFYZIOEQ
|
6.8 | IC50 | 2 | — | |
YLWSVZLNZZVTSM
|
6.8 | IC50 | 15 | — | |
IXDIKQYUVPRTQH
|
6.8 | IC50 | 6 | — | |
KXJILSLZMSOTHK
|
6.8 | IC50 | 6 | — | |
MCHFBGTXGSLCLO
|
6.8 | IC50 | 2 | — | |
MGXMGVUPCOMEOS
|
6.8 | IC50 | 5 | — | |
NYDBQVDGDFSUFN
|
6.8 | IC50 | 4 | — | |
WNYMMGOZYJKIQP
|
6.8 | IC50 | 4 | — | |
GIKCRZBMUUSXRT
|
6.8 | IC50 | 2 | — | |
HFDRYTOEWXVZHD
|
6.8 | IC50 | 2 | — | |
JOPRFEFNCAOJIR
|
6.8 | IC50 | 2 | — | |
QQWJGOWPTXJPPN
|
6.8 | IC50 | 2 | — | |
XBDBJEAKPCJTPF
|
6.8 | IC50 | 2 | — | |
CKVXYSBVFGGCGL
|
6.7 | IC50 | 5 | — | |
ORRPNEOZKXOAFX
|
6.7 | Ki | 4 | — | |
CQXYAWGSQLDRAK
|
6.7 | IC50 | 3 | — | |
FLIVKVQMXOAQAK
|
6.7 | IC50 | 15 | — | |
URGUVOCQHNXEMK
|
6.7 | IC50 | 2 | — | |
XGRCNZHEALOUNS
|
6.7 | IC50 | 2 | — | |
ASGMFNBUXDJWJJ
|
6.7 | IC50 | 8 | — | |
VEPOCTYIFBFDRZ
|
6.7 | IC50 | 4 | — | |
AUSDRYPYNGBOOX
|
6.7 | IC50 | 2 | — | |
FFQWDZFHWMXCGK
|
6.7 | IC50 | 5 | — | |
FFQWDZFHWMXCGK
|
6.7 | IC50 | 5 | — | |
FFVBCPCSHYDMLQ
|
6.7 | IC50 | 2 | — | |
HNUMRWMKXMAWTC
|
6.7 | IC50 | 2 | — | |
LHMJTCJXGOQGEX
|
6.7 | IC50 | 6 | — | |
ORKAKWRVOOOMDD
|
6.7 | IC50 | 4 | — | |
PHVGAEJTLZFYTO
|
6.7 | IC50 | 11 | — | |
TVZKWMUWNDZPCZ
|
6.7 | IC50 | 2 | — | |
ZASLFNNBUMDNJF
|
6.7 | IC50 | 2 | — | |
MQSVIANYXKTUMS
|
6.7 | IC50 | 2 | — | |
CWGKHYILSMYODL
|
6.7 | IC50 | 2 | — | |
GYGIXVNDVQQAPJ
|
6.7 | IC50 | 4 | — | |
MRPGRAKIAJJGMM
|
6.7 | IC50 | 11 | — |