Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIHKTGDJUXUJMJ
|
6.9 | IC50 | 4 | — | |
ZXNKLLQATJHCGU
|
6.9 | IC50 | 2 | — | |
DAAIOFDFLWLJLR
|
6.9 | IC50 | 2 | — | |
DEIFYFMWJVRUHV
|
6.9 | IC50 | 2 | — | |
IRQBQPNOWKSJBR
|
6.9 | IC50 | 2 | — | |
BTGKONUBBUHPMC
|
6.9 | IC50 | 2 | — | |
JUCHGYUYTUMHRL
|
6.9 | IC50 | 2 | — | |
QRFNPZUNAUBFQC
|
6.9 | IC50 | 4 | — | |
ULNHPTFPYSEATR
|
6.9 | IC50 | 2 | — | |
CELCCCWTAADGDV
|
6.9 | IC50 | 15 | — | |
PKCRUPNVGJBRRJ
|
6.9 | Ki | 4 | — | |
WTWMNNKZEVJCBK
|
6.9 | IC50 | 5 | — | |
GJVQDJDRGASLPK
|
6.9 | Ki | 4 | — | |
HZABJFRMYVCNTG
|
6.9 | IC50 | 4 | — | |
ICCWQZQHILTVNE
|
6.9 | Ki | 4 | — | |
KFRGPUFONMCXQI
|
6.9 | IC50 | 11 | — | |
LTJSYFAVWOFESN
|
6.9 | Ki | 4 | — | |
QNTSWLKVCFHNLY
|
6.9 | IC50 | 2 | — | |
VCHBBLKMWHUOMF
|
6.9 | IC50 | 2 | — | |
ILCHKGHOAZIHFP
|
6.9 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.9 | IC50 | 85 | Yes | |
RRJNXBNVQSVJBA
|
6.9 | IC50 | 2 | — | |
URASAXYDDZARND
|
6.9 | IC50 | 2 | — | |
WFAWAQUXUURRFW
|
6.9 | IC50 | 2 | — | |
YVGUVHSVOMWPCR
|
6.9 | Ki | 4 | — | |
JYRRTOFZIGEMAN
|
6.9 | IC50 | 2 | — | |
RGHJAGUBWMVUKC
|
6.9 | IC50 | 2 | — | |
SDRUQGPFTWNIMT
|
6.9 | IC50 | 2 | — | |
SHEPFXMPLORKLW
|
6.9 | Ki | 8 | — | |
GGCGIJHMDOQYGZ
|
6.9 | IC50 | 2 | — | |
NNARRPXFHVYBGW
|
6.9 | Ki | 4 | — | |
CEIJSVLEARLWRF
|
6.9 | IC50 | 13 | — | |
HOHCIMWLYQWLHB
|
6.9 | IC50 | 2 | — | |
NZVIEGVPMXNSJT
|
6.9 | IC50 | 2 | — | |
VIWQLUWKBPPTGG
|
6.9 | IC50 | 2 | — | |
ZPOSVRUJUALHAX
|
6.9 | IC50 | 2 | — | |
BAFFTSARAOAHFW
|
6.8 | IC50 | 2 | — | |
CGMYNNHQYROWEE
|
6.8 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
6.8 | Kd | 97 | Yes | |
OUSFTKFNBAZUKL
|
6.8 | Kd | 58 | Yes | |
VOZSBSGPEIZDAJ
|
6.8 | IC50 | 2 | — | |
LLMKBTGLZJIAMY
|
6.8 | IC50 | 5 | — | |
SDQPABOSBRYYPV
|
6.8 | IC50 | 2 | — | |
ZAEJFWCQZAIGKP
|
6.8 | IC50 | 2 | — | |
CLUCXVSOAQMMRQ
|
6.8 | IC50 | 2 | — | |
GEFYRVKALMUFSB
|
6.8 | IC50 | 2 | — | |
KJHOORCYJSBANN
|
6.8 | IC50 | 15 | — | |
QKWVFUHMEVWTPU
|
6.8 | IC50 | 2 | — | |
FKAJEPVSQITQLJ
|
6.8 | IC50 | 15 | — | |
HPSQCNGDSWWUNK
|
6.8 | IC50 | 2 | — |