Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AXNAPVYCQOKPOV
|
7.0 | IC50 | 2 | — | |
GLXOBAUWZZUWAU
|
7.0 | IC50 | 2 | — | |
NEXSFQXPWRMTDB
|
7.0 | IC50 | 2 | — | |
OKIKSBCVNZBYGX
|
7.0 | IC50 | 5 | — | |
PTKMSTJCOJHQGV
|
7.0 | Ki | 6 | — | |
WAOFSGJFQLXAOO
|
7.0 | IC50 | 2 | — | |
UYJPNAFIWZUXNS
|
7.0 | IC50 | 2 | — | |
AZMDWSWKDPCSEA
|
7.0 | Ki | 4 | — | |
BDEBDRHFGKUMKB
|
7.0 | IC50 | 2 | — | |
BKOOLLRJJOFPDK
|
7.0 | IC50 | 2 | — | |
CUOAKASSZZNNNL
|
7.0 | IC50 | 2 | — | |
CVNFODJWDVMZMH
|
7.0 | IC50 | 2 | — | |
DCYVUTFLZDIIOF
|
7.0 | IC50 | 2 | — | |
DWEDKXYEDVRUPT
|
7.0 | IC50 | 2 | — | |
GGIKBADETXOZQN
|
7.0 | IC50 | 2 | — | |
GKOZSLFVXRACHA
|
7.0 | IC50 | 3 | — | |
HHJFKJWFTARPJK
|
7.0 | IC50 | 3 | — | |
IVKDOOFDSADYOE
|
7.0 | IC50 | 3 | — | |
JEMUKTFLVUMJMN
|
7.0 | IC50 | 2 | — | |
JWENCJQYRRLPDS
|
7.0 | IC50 | 2 | — | |
LIMCXPZKZDPKPE
|
7.0 | IC50 | 2 | — | |
LJGDIIUPZAUEAC
|
7.0 | IC50 | 2 | — | |
LLRBNEGIXXRGLP
|
7.0 | Ki | 4 | — | |
LURAKVXKLBZZAP
|
7.0 | IC50 | 2 | — | |
MCGYAQRNWYNCMH
|
7.0 | IC50 | 2 | — | |
NHRSVTGGIGHXBM
|
7.0 | IC50 | 2 | — | |
QAIJLXROJVFNMR
|
7.0 | IC50 | 2 | — | |
QDTMPQOORBQFIG
|
7.0 | IC50 | 5 | — | |
QENIZOBYSVBQMH
|
7.0 | IC50 | 2 | — | |
QSZSUKPGDBYGQJ
|
7.0 | IC50 | 2 | — | |
SCUQJCIFMRPJSF
|
7.0 | IC50 | 2 | — | |
SGEWLDOMXQQVDJ
|
7.0 | IC50 | 3 | — | |
UDJDPLRKMXFFHF
|
7.0 | IC50 | 2 | — | |
URTMWTKJLRDYRH
|
7.0 | IC50 | 2 | — | |
VRSPEIRDNLLDBS
|
7.0 | IC50 | 2 | — | |
WFRGJVMNASTFDG
|
7.0 | IC50 | 2 | — | |
WVZHIWKRRWPURP
|
7.0 | IC50 | 2 | — | |
YSGSQQUJYWOWGW
|
7.0 | IC50 | 2 | — | |
YVPQULSHNCBRGY
|
7.0 | IC50 | 3 | — | |
YZXROTWIEAUPOA
|
7.0 | IC50 | 2 | — | |
DFTOONDZZWJTIX
|
7.0 | IC50 | 2 | — | |
GTVWYIASBVPCEA
|
7.0 | IC50 | 2 | — | |
JESGKYVOWCEUEO
|
7.0 | IC50 | 2 | — | |
JQOIYKPXKQECLH
|
7.0 | IC50 | 2 | — | |
KZLAQACITMZMTD
|
7.0 | IC50 | 2 | — | |
MLYXNIOIRSBOLQ
|
7.0 | IC50 | 2 | — | |
UNSAZGGWYRHTHJ
|
7.0 | IC50 | 3 | — | |
WAPRNUXTJDENKW
|
7.0 | IC50 | 2 | — | |
YQFQTKOIKKIREQ
|
7.0 | IC50 | 2 | — | |
ATWZRMIJXKDYLD
|
6.9 | Ki | 4 | — |