Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VVPJJCCYVVBFLO
|
7.1 | Ki | 4 | — | |
XRAHIDZAOGSWBC
|
7.1 | IC50 | 4 | — | |
JXKYPLVWZPUCOD
|
7.1 | IC50 | 2 | — | |
MMHOKKKPDYDUDS
|
7.1 | Ki | 4 | — | |
MSIYPAKNNNBUFM
|
7.1 | IC50 | 3 | — | |
RWSCYFXGWJPUQX
|
7.1 | IC50 | 15 | — | |
CLJQWNJQMODFSC
|
7.1 | IC50 | 2 | — | |
HXRJRZOYIVDQKX
|
7.1 | IC50 | 2 | — | |
PYCWIYZCNJUCBP
|
7.1 | Ki | 4 | — | |
SYAWYERBYBTWAB
|
7.1 | IC50 | 2 | — | |
ZINMQNQKXGNWQN
|
7.1 | IC50 | 2 | — | |
GULUZCYKKDJDGN
|
7.1 | IC50 | 3 | — | |
QTIXYWRLCYOCRY
|
7.1 | IC50 | 2 | — | |
XGOMMKURQRBZIA
|
7.1 | IC50 | 2 | — | |
IYZMPNPKBTXSTR
|
7.0 | IC50 | 3 | — | |
KQKZAECPRODPBM
|
7.0 | IC50 | 3 | — | |
LSCLFKMMDSPABA
|
7.0 | IC50 | 5 | — | |
NNNILSWONKWIJC
|
7.0 | Ki | 4 | — | |
QKGQVNUHCXZGQO
|
7.0 | IC50 | 2 | — | |
VSVLGWWGGFOSTP
|
7.0 | Ki | 4 | — | |
KCVLUTIUWHAOLI
|
7.0 | IC50 | 2 | — | |
FSCDYKUUMJNPMN
|
7.0 | IC50 | 2 | — | |
JLKCRZPBMOKDEB
|
7.0 | IC50 | 2 | — | |
KSCSDVHAZVSGAW
|
7.0 | Ki | 4 | — | |
MSCWTVCDJKKGHK
|
7.0 | Ki | 4 | — | |
ONRJNVZFOSHIQI
|
7.0 | Ki | 8 | — | |
UYRUSUBNRZEGRJ
|
7.0 | IC50 | 2 | — | |
VCVZEWLIGPYLQF
|
7.0 | IC50 | 2 | — | |
BIQADQASLLQRRS
|
7.0 | IC50 | 2 | — | |
CVBIOKGKBZUACK
|
7.0 | IC50 | 2 | — | |
GLDVFVXCMSQZMZ
|
7.0 | IC50 | 4 | — | |
IAPISFUJUUDVNW
|
7.0 | IC50 | 15 | — | |
KWTCGLLOWQHMIN
|
7.0 | IC50 | 2 | — | |
QKWHDVWGAMZGHO
|
7.0 | Ki | 4 | — | |
CNNOAGXHCAVQKZ
|
7.0 | IC50 | 13 | — | |
FHMFHOQHUFKWBK
|
7.0 | IC50 | 3 | — | |
HCDMSNJPLKSFOG
|
7.0 | Ki | 4 | — | |
HDKIHQOXUMCGPU
|
7.0 | Ki | 6 | — | |
IELILXSXGFXHAH
|
7.0 | IC50 | 2 | — | |
MIJLYWBJXSCQRT
|
7.0 | IC50 | 2 | — | |
PTMIZOWGQFVIPS
|
7.0 | IC50 | 2 | — | |
QKUPEYVJRBJWLO
|
7.0 | IC50 | 6 | — | |
RYPUWZOEFAAXRB
|
7.0 | IC50 | 6 | — | |
SNMMJBCMTCRCSM
|
7.0 | IC50 | 13 | — | |
BBDLGEJJPNXUSB
|
7.0 | IC50 | 4 | — | |
COWADZBACSGMBW
|
7.0 | IC50 | 2 | — | |
FIQBYSRAADOZQW
|
7.0 | Ki | 4 | — | |
HRCYPBKRTCCYMF
|
7.0 | IC50 | 2 | — | |
NSWBUBCIZVPAIF
|
7.0 | IC50 | 2 | — | |
WUPRAHSNJBLKQZ
|
7.0 | IC50 | 2 | — |