Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BJYQLWPTBHMZKP
|
7.2 | IC50 | 5 | — | |
GGTPTLANFCGFPU
|
7.2 | IC50 | 8 | — | |
KTAKVDASVPBVHO
|
7.2 | IC50 | 2 | — | |
DFQHKYRGJBTDLZ
|
7.2 | IC50 | 3 | — | |
TYSWNLQZLBRNSE
|
7.2 | IC50 | 15 | — | |
XMTXXRRXTXBUMH
|
7.2 | IC50 | 2 | — | |
YZANXEFHQOKRIL
|
7.2 | Ki | 4 | — | |
ZSHKDJHZNZUYQM
|
7.2 | IC50 | 3 | — | |
UIAYOLLUEZBQEH
|
7.2 | IC50 | 6 | — | |
UNVBFURIHRAGGO
|
7.2 | Ki | 6 | — | |
YWCRCIBLGLRDHR
|
7.2 | IC50 | 2 | — | |
FCWICHXUWNYHMX
|
7.2 | IC50 | 4 | — | |
KOSUFZUQHXDTAI
|
7.2 | IC50 | 5 | — | |
XDLFXLIRQNNHLS
|
7.2 | IC50 | 2 | — | |
YHKQITMSINAKOO
|
7.2 | IC50 | 3 | — | |
ZDJLCMWGZIMCAQ
|
7.2 | Ki | 4 | — | |
ZFOXIJRTZOAGDX
|
7.2 | IC50 | 4 | — | |
JBNYXSCCYVQNFW
|
7.2 | IC50 | 2 | — | |
SBKJAWVXVBLZEB
|
7.2 | IC50 | 2 | — | |
URASAXYDDZARND
|
7.2 | IC50 | 2 | — | |
CCYFCUHYFHNQAO
|
7.2 | IC50 | 3 | — | |
KLVYMYQTRZCMLE
|
7.2 | IC50 | 11 | Yes | |
HKVDMDVJPHFROE
|
7.1 | IC50 | 2 | — | |
DHRDOFYSAXLFOH
|
7.1 | IC50 | 2 | — | |
OVRDWLJZSQZCBW
|
7.1 | IC50 | 2 | — | |
POVOYMIAJXXYSA
|
7.1 | IC50 | 3 | — | |
AFPVWMUZKWPINC
|
7.1 | IC50 | 2 | — | |
DQBKPGGGGXRALY
|
7.1 | IC50 | 4 | — | |
LBCPIVDSZHGQAB
|
7.1 | IC50 | 3 | — | |
NUPYFDZMVCSJTN
|
7.1 | IC50 | 2 | — | |
OYRHVLHXZXDTIQ
|
7.1 | IC50 | 2 | — | |
UMSHWYWDNHHQIT
|
7.1 | IC50 | 2 | — | |
VAXZNXSXFNHQFE
|
7.1 | IC50 | 3 | — | |
WOSWUKXUZVAPGM
|
7.1 | IC50 | 3 | — | |
YNOMJXFCXSQSEU
|
7.1 | IC50 | 3 | — | |
ZMXFWVYPMCRPSG
|
7.1 | IC50 | 3 | — | |
ZNHOBBHQPZULFS
|
7.1 | IC50 | 3 | — | |
ZPHBEDTYTQWLFC
|
7.1 | IC50 | 13 | — | |
ZWXBEUSAAVHLFW
|
7.1 | IC50 | 8 | — | |
AREQVYHOGWNDNY
|
7.1 | IC50 | 2 | — | |
BVVBONNOUZEEBK
|
7.1 | IC50 | 2 | — | |
IWXGANKLKSELIX
|
7.1 | IC50 | 2 | — | |
QOFBRKYUXYHDLI
|
7.1 | Ki | 4 | — | |
RLAAXHAIRXSBGB
|
7.1 | IC50 | 3 | — | |
BIIVYFLTOXDAOV
|
7.1 | IC50 | 82 | Yes | |
IADNEAHKTOVOBX
|
7.1 | IC50 | 4 | — | |
NSFWLIYQFQEQDW
|
7.1 | IC50 | 6 | — | |
KSCSDVHAZVSGAW
|
7.1 | Ki | 4 | — | |
MIFCTDCDIAKSQG
|
7.1 | Ki | 6 | — | |
PJJINEFZNAWLHB
|
7.1 | Ki | 4 | — |