Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QCBLVLKFDWENOV
|
7.3 | IC50 | 4 | — | |
QMXSDPDZRQFBHB
|
7.3 | IC50 | 5 | — | |
QUWHYVIAUBWWFO
|
7.3 | IC50 | 4 | — | |
QWNPBVNMKNDQGI
|
7.3 | IC50 | 5 | — | |
RHMBFFCPOJVSLV
|
7.3 | Ki | 4 | — | |
RTOZTQPNHKYMFF
|
7.3 | IC50 | 3 | — | |
SBNVUFMJQUOIKN
|
7.3 | IC50 | 9 | — | |
SMJQEMBROAGZDG
|
7.3 | IC50 | 4 | — | |
SZDWEMLCKOXDFZ
|
7.3 | IC50 | 3 | — | |
TXBBMRZBMVLLAQ
|
7.3 | IC50 | 6 | — | |
TYCIGEQMTDJQIM
|
7.3 | IC50 | 5 | — | |
TZUUUOFIEZNZEI
|
7.3 | IC50 | 4 | — | |
UAAXTVOYMWPDBQ
|
7.3 | IC50 | 6 | — | |
VBLLOFSUFOWCAN
|
7.3 | IC50 | 6 | — | |
VBTFDZNKWVGQPG
|
7.3 | IC50 | 6 | — | |
VEZGUWKKHGUXIU
|
7.3 | IC50 | 5 | — | |
WGPONUKJUHDRKT
|
7.3 | IC50 | 3 | — | |
WNPAEAQXLNHGQL
|
7.3 | IC50 | 6 | — | |
XNTXGZBBRXIZGX
|
7.3 | IC50 | 3 | — | |
XSIFHJZCEOMGNC
|
7.3 | IC50 | 4 | — | |
YFUMBTADPXPQKL
|
7.3 | Ki | 4 | — | |
YOHCMXQAXUTESC
|
7.3 | IC50 | 5 | — | |
ZIWFXQFVSGOWAZ
|
7.3 | Ki | 6 | — | |
ZWWQVYKYWCWYFJ
|
7.3 | IC50 | 5 | — | |
GFXPNXYGBQGEGI
|
7.2 | Ki | 4 | — | |
IUNFVCUQVDDZRS
|
7.2 | IC50 | 2 | — | |
PJMQGCMGADZNSF
|
7.2 | Ki | 4 | — | |
IXCNPHLUEWEYKF
|
7.2 | IC50 | 3 | — | |
KMVBIPSQSSTTCJ
|
7.2 | IC50 | 11 | — | |
MAZYMHDZBKSRMW
|
7.2 | IC50 | 2 | — | |
QKFMIXAVODWZLI
|
7.2 | IC50 | 2 | — | |
UKLWPHGHSYZRHP
|
7.2 | IC50 | 2 | — | |
UTHWBIPHRYUJSU
|
7.2 | IC50 | 11 | Yes | |
XJPIUXVIFQKKQE
|
7.2 | Ki | 4 | — | |
YGFJSPTVMIFQBT
|
7.2 | IC50 | 2 | — | |
GJYFUNGTPLHRJF
|
7.2 | IC50 | 2 | — | |
IJIGRXABGQBDBA
|
7.2 | Ki | 10 | — | |
QYJLBHRAPDJOSO
|
7.2 | Ki | 4 | — | |
ULLGENQITYAYQU
|
7.2 | IC50 | 2 | — | |
BGYGYQGUFXBQFT
|
7.2 | IC50 | 2 | — | |
FDOSHYORLAUOGZ
|
7.2 | IC50 | 2 | — | |
GEHWYWMDTGSDFR
|
7.2 | Ki | 4 | — | |
JBWJGEZTYVAWBR
|
7.2 | IC50 | 2 | — | |
MRBRAJMKQXXCBZ
|
7.2 | IC50 | 2 | — | |
ONESBFJNZYJCEA
|
7.2 | IC50 | 2 | — | |
PFWXLZFOFFJJKK
|
7.2 | IC50 | 2 | — | |
PTMADKDGOQDQEW
|
7.2 | IC50 | 2 | — | |
PZNJKWXGJKXLOU
|
7.2 | IC50 | 4 | — | |
WCYXZWGSJXHMPW
|
7.2 | IC50 | 2 | — | |
ZISIZBLHDWUJIQ
|
7.2 | IC50 | 2 | — |