Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MRYLLITXXQUJLZ
|
7.4 | IC50 | 5 | — | |
PDJVJMYVUAQPLU
|
7.4 | IC50 | 3 | — | |
QFTKYJVUSSEJCS
|
7.4 | IC50 | 4 | — | |
QIQHZHDHJRCDDH
|
7.4 | IC50 | 2 | — | |
UBHPJEJMHASIRC
|
7.4 | IC50 | 6 | — | |
XDDTXXUNFPYDOF
|
7.4 | IC50 | 2 | — | |
GBYGWVVFPYTZJX
|
7.4 | IC50 | 4 | — | |
LKRBWJATDRLWCK
|
7.4 | IC50 | 2 | — | |
RSJIUPFUDJRJNK
|
7.4 | Ki | 4 | — | |
XYZIPKBTOPMPRH
|
7.4 | IC50 | 4 | — | |
DSNLTPDDMYUGMH
|
7.4 | IC50 | 2 | — | |
HTBKVAJZYRVZSW
|
7.4 | IC50 | 11 | — | |
RHESBWSFHDYVKX
|
7.4 | Ki | 4 | — | |
FKAJEPVSQITQLJ
|
7.3 | IC50 | 15 | — | |
NFTJDXGFOUFNKG
|
7.3 | IC50 | 16 | — | |
NOJFQFRTLNURFX
|
7.3 | IC50 | 2 | — | |
ONCJKEZPQVEATH
|
7.3 | IC50 | 2 | — | |
RDLLMXCIBZYDEZ
|
7.3 | IC50 | 2 | — | |
TTZAURANQVEMPE
|
7.3 | IC50 | 4 | — | |
VAPFBPVHSQVGMQ
|
7.3 | Ki | 4 | — | |
DHQOXLRGBCLMFX
|
7.3 | IC50 | 2 | — | |
KRRAKMWTYZXXLV
|
7.3 | IC50 | 2 | — | |
PQTGAAIDDFNDPD
|
7.3 | IC50 | 4 | — | |
QCMQTRDINCHRHG
|
7.3 | Ki | 4 | — | |
UBYXZTIDJPASEM
|
7.3 | IC50 | 2 | — | |
UDBGEYDMPMCZES
|
7.3 | IC50 | 2 | — | |
XONPCCFQRCPXJB
|
7.3 | IC50 | 3 | — | |
FLNHSHVOGZEONH
|
7.3 | IC50 | 4 | — | |
LQOVXXQVZQEEKA
|
7.3 | IC50 | 6 | — | |
DIFUHKJZJNRRMN
|
7.3 | IC50 | 9 | — | |
VGPGCCHHKHQDOQ
|
7.3 | IC50 | 2 | — | |
ZFPLWUCEDGLIET
|
7.3 | IC50 | 2 | — | |
IIIIVBPOQAVFDM
|
7.3 | IC50 | 2 | — | |
PNLPHGXRRNXSNB
|
7.3 | IC50 | 11 | — | |
POJGZHZSQVZDGP
|
7.3 | IC50 | 7 | — | |
XPWRDXLMZNJXQQ
|
7.3 | Ki | 4 | — | |
BEFVJTSMLGHNEY
|
7.3 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.3 | IC50 | 408 | — | |
NQDANZVBQUDPGE
|
7.3 | Ki | 4 | — | |
UTSBHEVQCONLCR
|
7.3 | IC50 | 4 | — | |
VBKQQDIWFTTXHE
|
7.3 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
7.3 | IC50 | 46 | — | |
CGMYNNHQYROWEE
|
7.3 | IC50 | 2 | — | |
CXMKIWPGGSLHRE
|
7.3 | IC50 | 15 | — | |
FCZVSNICWQFRLO
|
7.3 | Ki | 4 | — | |
NMEUNCBNBWJJFA
|
7.3 | Ki | 4 | — | |
UVNWLDYNLOHPKC
|
7.3 | IC50 | 5 | — | |
AUARWWSRHMPTLW
|
7.3 | IC50 | 3 | — | |
CCBZMLZJNJSZDY
|
7.3 | IC50 | 2 | — | |
FAMZJTKFGMSFPP
|
7.3 | IC50 | 3 | — |