Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KXFIUSMEECFBBN
|
7.4 | Ki | 4 | — | |
NBSJZWFDNFWQDN
|
7.4 | IC50 | 29 | — | |
OYOOKQHAKAOWPK
|
7.4 | IC50 | 2 | — | |
PNPPYTKHXUSEOA
|
7.4 | IC50 | 5 | — | |
RONAHISFEVHOEE
|
7.4 | IC50 | 8 | — | |
VXNBBAUTPXCUOZ
|
7.4 | IC50 | 2 | — | |
WURCEOZSLIZNTF
|
7.4 | IC50 | 2 | — | |
WVMNAFHMDQOKIP
|
7.4 | IC50 | 4 | — | |
XVUSHGLGCAFDEU
|
7.4 | Ki | 4 | — | |
AVLXLHMRMWGCNQ
|
7.4 | IC50 | 2 | — | |
CPTPRZGRXQWAQQ
|
7.4 | Ki | 4 | — | |
FOPZTCDUAPTHJY
|
7.4 | IC50 | 4 | — | |
GVAFORCHGQCAGW
|
7.4 | IC50 | 3 | — | |
JZBKRUVPRZMVNL
|
7.4 | IC50 | 4 | — | |
MRCKOWVLVZNAPU
|
7.4 | IC50 | 2 | — | |
MSPNNLMRAHNGBB
|
7.4 | IC50 | 3 | — | |
NDJJMTZAXWRELC
|
7.4 | IC50 | 2 | — | |
XPMRMPBWKVMUTB
|
7.4 | Ki | 5 | — | |
ZEWYBLWRWWDFIL
|
7.4 | IC50 | 3 | — | |
DNYGSWNXJXELOX
|
7.4 | Ki | 5 | — | |
GGRSBRWNHVOEPC
|
7.4 | IC50 | 2 | — | |
HLUPUMQWJOFHGU
|
7.4 | IC50 | 2 | — | |
HMBBGEYXFQLFSV
|
7.4 | IC50 | 2 | — | |
LURUBKPSGYTVJA
|
7.4 | IC50 | 3 | — | |
PUWXPMFEDYRLTM
|
7.4 | IC50 | 6 | — | |
QVZHUFDUPLWTFU
|
7.4 | Ki | 4 | — | |
WFRQTWKTDYNOMW
|
7.4 | IC50 | 2 | — | |
ZEKYDJPVMYFVGA
|
7.4 | IC50 | 2 | — | |
COHWLZJUNHSLBR
|
7.4 | Ki | 4 | — | |
QULVCQWDONFUCP
|
7.4 | IC50 | 2 | — | |
RHXHGRAEPCAFML
|
7.4 | IC50 | 9 | — | |
SKOICOFQIQHEPE
|
7.4 | IC50 | 9 | — | |
VXZRTFJMWFQYND
|
7.4 | Ki | 4 | — | |
WTYQQWZPWDYEMU
|
7.4 | IC50 | 2 | — | |
WWUPNOVYRXPGJZ
|
7.4 | IC50 | 5 | — | |
DNVODRITWXGBQB
|
7.4 | IC50 | 4 | — | |
GIDODEPBXGRWBW
|
7.4 | IC50 | 2 | — | |
GIDODEPBXGRWBW
|
7.4 | IC50 | 2 | — | |
IGFRKWYWGSYHGA
|
7.4 | IC50 | 5 | — | |
JYVQQVITMQSABB
|
7.4 | IC50 | 2 | — | |
NKSJUACUARPPLH
|
7.4 | IC50 | 13 | — | |
SFFBXSHJSYMDGI
|
7.4 | Ki | 4 | — | |
UYSQOPXDZOJYOF
|
7.4 | IC50 | 2 | — | |
YJBGQSYONUDUCN
|
7.4 | Ki | 3 | — | |
NBJSISKLAZWALR
|
7.4 | IC50 | 2 | — | |
QVTBPKJVDXGPQL
|
7.4 | IC50 | 5 | — | |
RECJWFRRTNLZDX
|
7.4 | Ki | 4 | — | |
VHWUUBMRANHHCU
|
7.4 | IC50 | 2 | — | |
XNFJUHZLDMOZHP
|
7.4 | IC50 | 2 | — | |
BASWGBOBVOPWNF
|
7.4 | IC50 | 4 | — |