Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPCNFXQXVGAXIF
|
7.5 | IC50 | 2 | — | |
PRGZEWRXEYVMGW
|
7.5 | Ki | 4 | — | |
QTEXRPQBMDQPDE
|
7.5 | IC50 | 11 | — | |
RMLWTYYGKGDCFZ
|
7.5 | IC50 | 4 | — | |
RVKNONNXSNALJV
|
7.5 | IC50 | 21 | — | |
UKVZKVRVVNTCMR
|
7.5 | Ki | 4 | — | |
WIINVKDUAJXWIM
|
7.5 | IC50 | 8 | — | |
XOJPAVACYRFOBK
|
7.5 | IC50 | 7 | — | |
IPALDEQYNHHIED
|
7.5 | IC50 | 2 | — | |
JWYHKDMZXSHNLA
|
7.5 | IC50 | 6 | — | |
PIMQWRZWLQKKBJ
|
7.5 | Kd | 36 | — | |
QCALUKUBCRTVRC
|
7.5 | Ki | 4 | — | |
RBMBLJOYIGVBNO
|
7.5 | IC50 | 6 | — | |
UKSFDLFTRMYZGG
|
7.5 | Ki | 5 | — | |
UQVXBLAVQKBUCD
|
7.5 | IC50 | 3 | — | |
LHEKUPICAYEUEL
|
7.5 | Ki | 4 | — | |
DCHQNZAIUFIFEB
|
7.5 | IC50 | 3 | — | |
FRUDYEUOYPWKKU
|
7.5 | IC50 | 5 | — | |
IPDNYZDGHMOFHG
|
7.5 | IC50 | 2 | — | |
OQEFZDKDXVHSRX
|
7.5 | IC50 | 4 | — | |
QDOVUCKBHKKVRH
|
7.5 | IC50 | 2 | — | |
QYUAZFYQXCJXEM
|
7.5 | IC50 | 3 | — | |
SZRNZUUUCFGQSQ
|
7.5 | IC50 | 2 | — | |
YXBKCKHBHRIXQX
|
7.5 | IC50 | 2 | — | |
BIEUJMYBFCQBTJ
|
7.5 | Ki | 4 | — | |
CGMQFXGWSKCKSF
|
7.5 | IC50 | 2 | — | |
IEYXXFUMUXPXFO
|
7.5 | Ki | 4 | — | |
JSMQRWBYWSIQRV
|
7.5 | IC50 | 2 | — | |
JTZWTKLEXMYEMU
|
7.5 | Ki | 6 | — | |
LAQCQSKKZIRXFW
|
7.5 | IC50 | 9 | — | |
LICNBVSSOUPXNB
|
7.5 | IC50 | 2 | — | |
MDMZHXGVQNUOHL
|
7.5 | Ki | 4 | — | |
OCPZYMHKJYHDEO
|
7.5 | IC50 | 2 | — | |
ORNZIPBQHSHKDI
|
7.5 | IC50 | 2 | — | |
RAFISFVOOKCYLW
|
7.5 | IC50 | 6 | — | |
SYAHGEVTXVOAGT
|
7.5 | IC50 | 3 | — | |
BNNYAWQVSWARTD
|
7.5 | IC50 | 3 | — | |
FPYTVDRQKLOFIJ
|
7.5 | IC50 | 2 | — | |
GCACFLIUQWTSKF
|
7.5 | IC50 | 3 | — | |
GITJQMOEQGGXTM
|
7.5 | IC50 | 3 | — | |
GKCCTOCVAIDPIB
|
7.5 | IC50 | 3 | — | |
IOQSBRPAWCWDTI
|
7.5 | IC50 | 3 | — | |
LFEZAGQLYZHSRW
|
7.5 | IC50 | 2 | — | |
NQVNNPOALMGCQC
|
7.5 | IC50 | 3 | — | |
RBVKWCPDHUGWQM
|
7.5 | IC50 | 3 | — | |
UUNRKBQEUSFVRI
|
7.5 | IC50 | 2 | — | |
WJCPRQRDANGIJZ
|
7.5 | IC50 | 3 | — | |
ZNYIGYODHSKJEZ
|
7.5 | IC50 | 3 | — | |
SMJIOBIBQNQQMH
|
7.5 | Ki | 4 | — | |
BAMUDEHGCAVPNN
|
7.4 | IC50 | 2 | — |