Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLFOYPRDIYQCLG
|
7.6 | IC50 | 2 | — | |
QCXMOVSRDNYGQN
|
7.6 | IC50 | 2 | — | |
UEQPGBQDKMIYEQ
|
7.6 | IC50 | 2 | — | |
WBMDZLSDTLNSBE
|
7.6 | Ki | 4 | — | |
XKZZWESLMRHCAW
|
7.6 | IC50 | 5 | — | |
AZBVCCPKEJNWJE
|
7.6 | IC50 | 3 | — | |
BAZFEYHRFTWKSE
|
7.6 | Ki | 4 | — | |
CUOAKASSZZNNNL
|
7.6 | IC50 | 2 | — | |
JCRIMVWZWOWOPT
|
7.6 | IC50 | 2 | — | |
KNYGWCOOEMGKAK
|
7.6 | Ki | 4 | — | |
MAVGAHAOCLDZKW
|
7.6 | IC50 | 2 | — | |
NEEPJQJEJYVZAP
|
7.6 | IC50 | 2 | — | |
PFMKIDRZHBZULH
|
7.6 | IC50 | 6 | — | |
UJCYGTTWTLTIEZ
|
7.6 | IC50 | 5 | — | |
UXXXHEOMIMPLKB
|
7.6 | Ki | 4 | — | |
VCEVKRSWGMXHPO
|
7.6 | IC50 | 2 | — | |
YEHAPGDDUMGAOD
|
7.6 | IC50 | 2 | — | |
SGWSLLDTSFNPEK
|
7.6 | IC50 | 6 | — | |
ZKCDHUYJDPLBTG
|
7.6 | Ki | 4 | — | |
AJTMZFRCOLMNQV
|
7.5 | IC50 | 2 | — | |
AXODIUJQDFIKDJ
|
7.5 | IC50 | 2 | — | |
CAOFILCIPZJTLM
|
7.5 | IC50 | 4 | — | |
CGMYFNOVLBOMQH
|
7.5 | Ki | 4 | — | |
CGMYFNOVLBOMQH
|
7.5 | Ki | 4 | — | |
GDZVTFLLGJNTRE
|
7.5 | IC50 | 11 | — | |
HBUAOMASWHOWJB
|
7.5 | Ki | 8 | — | |
JJJVFTNNFDYRFZ
|
7.5 | IC50 | 2 | — | |
LGTNVNQWJQDILD
|
7.5 | IC50 | 5 | — | |
YCANTYAOGZQCIG
|
7.5 | IC50 | 2 | — | |
YNERHABIIHQUTQ
|
7.5 | IC50 | 2 | — | |
AWOBBZHRSADRLH
|
7.5 | IC50 | 2 | — | |
KDIKLUVXDINZHL
|
7.5 | IC50 | 4 | — | |
LVLNKVFDBFRZPR
|
7.5 | Ki | 4 | — | |
SOTUJCQXHVILHQ
|
7.5 | Ki | 4 | — | |
YECDMWPRVSKSOX
|
7.5 | IC50 | 4 | — | |
FXNYFKNNCUKUAE
|
7.5 | IC50 | 3 | — | |
DFRLATSJZFEZJT
|
7.5 | IC50 | 2 | — | |
FLELSIDTMCCIRQ
|
7.5 | IC50 | 2 | — | |
LPNUTFAGTQJSOJ
|
7.5 | Ki | 4 | — | |
LTQWMHQCZKPWSG
|
7.5 | IC50 | 2 | — | |
PPJRGLDUXCYWQR
|
7.5 | IC50 | 2 | — | |
PUHKAOLWMGXVFS
|
7.5 | IC50 | 3 | — | |
UGKFAPJXEKVBHI
|
7.5 | Ki | 4 | — | |
XJYHNBLHADKOIG
|
7.5 | IC50 | 2 | — | |
ZZUHVLBKVYTZJN
|
7.5 | IC50 | 2 | — | |
GYTNVEDSWNLDQV
|
7.5 | Ki | 6 | — | |
LCZLJATWTUPEBT
|
7.5 | IC50 | 2 | — | |
LDHMPOHMNQEDFG
|
7.5 | Ki | 4 | — | |
MENAPVXPHDXOTR
|
7.5 | IC50 | 2 | — | |
NVMQZCJPKNUECR
|
7.5 | IC50 | 2 | — |