Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IQPGVUQARGVQGU
|
7.6 | IC50 | 2 | — | |
JFIULCBZFIWZRF
|
7.6 | IC50 | 2 | — | |
JZGPEQNPASOUFO
|
7.6 | IC50 | 3 | — | |
KHDFBLMRVOKCMV
|
7.6 | IC50 | 2 | — | |
OBJNQQWSNUSMIU
|
7.6 | IC50 | 3 | — | |
OQAXDEGUMXXBQC
|
7.6 | IC50 | 2 | — | |
PFIWFAQPXJTVMJ
|
7.6 | IC50 | 3 | — | |
QELIOBZBBHRBAA
|
7.6 | Ki | 4 | — | |
QROLGGZKPDXPRM
|
7.6 | Ki | 4 | — | |
VMEQMRCCKBMZLT
|
7.6 | IC50 | 4 | — | |
VWHFRLLFAUDIJB
|
7.6 | Ki | 4 | — | |
DQLJIEVRWTVXIO
|
7.6 | Ki | 4 | — | |
KUXCGTVJRJBHEO
|
7.6 | Ki | 4 | — | |
USGHJKLVOOFHKH
|
7.6 | Ki | 4 | — | |
ZAFRFGKCOSNMCP
|
7.6 | Ki | 4 | — | |
FCIFHHREDAFKNR
|
7.6 | IC50 | 3 | — | |
JHSKWDLRXRYFOQ
|
7.6 | Ki | 4 | — | |
KBNBMEPJGLGMRS
|
7.6 | IC50 | 2 | — | |
QRVJVTAVMDZGBU
|
7.6 | IC50 | 8 | — | |
QYKOXFSITMBUDO
|
7.6 | IC50 | 2 | — | |
SMNBJOCPOYEKDE
|
7.6 | IC50 | 2 | — | |
UHKSQQNYPYARFR
|
7.6 | IC50 | 2 | — | |
VQBVWRIVPOILKH
|
7.6 | Ki | 3 | — | |
XNFJUHZLDMOZHP
|
7.6 | IC50 | 2 | — | |
YGMXOJBZAZZNRV
|
7.6 | IC50 | 2 | — | |
YMOIBDPPXWKGFR
|
7.6 | IC50 | 3 | — | |
YXNQYHXLQNMLSB
|
7.6 | IC50 | 5 | — | |
BPWNKOBNYHBQJR
|
7.6 | Ki | 4 | — | |
FJPAQWZAYUMSQZ
|
7.6 | Ki | 4 | — | |
HFCRZSDUGZDJHM
|
7.6 | IC50 | 2 | — | |
BIEUJMYBFCQBTJ
|
7.6 | Ki | 4 | — | |
BKJVBBWPOYUPFA
|
7.6 | IC50 | 2 | — | |
IMANTSACQRSZER
|
7.6 | IC50 | 2 | — | |
JBPAAOAEZFTBLA
|
7.6 | IC50 | 2 | — | |
OFTAQYQPSSRBOZ
|
7.6 | Ki | 4 | — | |
VAWYHOYAWTUTHR
|
7.6 | IC50 | 4 | — | |
WCEJWHANTHYYCV
|
7.6 | IC50 | 3 | — | |
YOZIUASNGGMFQI
|
7.6 | IC50 | 4 | — | |
AAYWXOINDKYXKL
|
7.6 | IC50 | 2 | — | |
FSSQAUUKDWDXEX
|
7.6 | Ki | 4 | — | |
KHUHONPSWMPDIC
|
7.6 | Ki | 4 | — | |
OFOKNGAIALWCMY
|
7.6 | IC50 | 2 | — | |
UZJAFJATSYCXRA
|
7.6 | IC50 | 3 | — | |
XZIQOSLQCRPOBS
|
7.6 | IC50 | 3 | — | |
ZFCILQSOMHMEON
|
7.6 | IC50 | 4 | — | |
AZXYPCBAGCXZPP
|
7.6 | IC50 | 4 | — | |
GKYNYPYSGJOBRE
|
7.6 | IC50 | 2 | — | |
HHFXMDZWCLHCFZ
|
7.6 | IC50 | 2 | — | |
JJDCFCXCIHINRQ
|
7.6 | IC50 | 5 | — | |
KRDTUJDAEVGZCU
|
7.6 | IC50 | 2 | — |