Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GJEWTVQXBHSVAU
|
7.7 | IC50 | 3 | — | |
GZUIGXOHHAYCLT
|
7.7 | IC50 | 6 | — | |
MCGRCAVMPSXODJ
|
7.7 | IC50 | 2 | — | |
XBOIHCUWWMWMIZ
|
7.7 | IC50 | 2 | — | |
AQRSMVCQDQNUQT
|
7.7 | IC50 | 2 | — | |
AYCUZAAKVCOJJW
|
7.7 | Ki | 4 | — | |
KABOFUDSOMJKKL
|
7.7 | Ki | 4 | — | |
ZAFRFGKCOSNMCP
|
7.7 | Ki | 4 | — | |
ZJASKMZRNIQJAD
|
7.7 | IC50 | 2 | — | |
CRHUKNBYXYKXBS
|
7.7 | IC50 | 2 | — | |
HWLTZCGRFYEWPQ
|
7.7 | IC50 | 2 | — | |
KHCQHSATOWGBMQ
|
7.7 | IC50 | 2 | — | |
NVGVEXRVOGUMEO
|
7.7 | Ki | 4 | — | |
SAWDJPCFUCEYJD
|
7.7 | Ki | 4 | — | |
SMNBJOCPOYEKDE
|
7.7 | IC50 | 2 | — | |
ULIMVSSEPMLVHV
|
7.7 | Ki | 6 | — | |
YPBVPXIBHMXSAS
|
7.7 | IC50 | 5 | — | |
HGINWKMFVVFJSI
|
7.7 | Ki | 4 | — | |
MVLOBPPFCUCBHT
|
7.7 | IC50 | 9 | — | |
RJOAAVPWGOLZSU
|
7.7 | IC50 | 2 | — | |
HMXNJXIHQSSEJY
|
7.7 | IC50 | 2 | — | |
JDUNFKKPNFKLEH
|
7.7 | IC50 | 2 | — | |
JGZXCZPRYTYKPZ
|
7.7 | IC50 | 2 | — | |
JXVCQGBDCQGWBV
|
7.7 | IC50 | 2 | — | |
JZLXIDIBRQZXJD
|
7.7 | IC50 | 2 | — | |
UHCMUGYUWQCODZ
|
7.7 | Ki | 5 | — | |
VTLCELVAADXYMP
|
7.7 | IC50 | 2 | — | |
WNBOZMLWGXPGLO
|
7.7 | IC50 | 2 | — | |
YHROUXCFDDZCJA
|
7.7 | IC50 | 3 | — | |
ZUUXXQZUHHHBPS
|
7.7 | IC50 | 2 | — | |
CGMYNNHQYROWEE
|
7.7 | IC50 | 2 | — | |
NXHNUMBGXRTEFE
|
7.7 | Ki | 4 | — | |
CMCOAKYYTHTADV
|
7.7 | Ki | 4 | — | |
DSSKUVUQTGKPGW
|
7.7 | IC50 | 2 | — | |
HFDVXFHTDRHDGR
|
7.7 | IC50 | 3 | — | |
JQDUGOIAGBCXFF
|
7.7 | IC50 | 3 | — | |
JRVLCPFGZSZGRN
|
7.7 | IC50 | 2 | — | |
MDFHINIKLRTFAE
|
7.7 | IC50 | 4 | — | |
SGOYVJDFFJKWDN
|
7.7 | IC50 | 2 | — | |
VGTZAEIJCBVBJN
|
7.7 | IC50 | 2 | — | |
WJRRGYBTGDJBFX
|
7.7 | IC50 | 16 | Yes | |
WSJLJBASYBSDMI
|
7.7 | IC50 | 2 | — | |
XJDGXENWWHQUCX
|
7.7 | IC50 | 2 | — | |
ZORUMGHLMKWRPP
|
7.7 | IC50 | 8 | — | |
AXTXGXVLRKZCFY
|
7.7 | Ki | 4 | — | |
BVZZSEVVEDNIOM
|
7.7 | IC50 | 3 | — | |
MJIIYXFGPPGPGB
|
7.7 | IC50 | 5 | — | |
PACLAQXDVXULPW
|
7.7 | Ki | 4 | — | |
VLWZGXZKJHXLTL
|
7.7 | IC50 | 3 | — | |
FQOMMDNBEIZMGZ
|
7.6 | Ki | 6 | — |