Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MDDQGEIMRPZKBT
|
7.8 | IC50 | 2 | — | |
NVJVPUYRSSDOPO
|
7.8 | IC50 | 2 | — | |
ORNZIPBQHSHKDI
|
7.8 | IC50 | 2 | — | |
POFVJRKJJBFPII
|
7.8 | Ki | 8 | — | |
UJLRCOLCMNEBIT
|
7.8 | IC50 | 2 | — | |
XDEIHTNJRRVHEQ
|
7.8 | IC50 | 5 | — | |
XFNINEDWLFKZMH
|
7.8 | IC50 | 3 | — | |
ZEKYDJPVMYFVGA
|
7.8 | IC50 | 2 | — | |
BBFMOOCYTUUCCR
|
7.8 | Ki | 4 | — | |
FTFMKZBZJAZXTH
|
7.8 | Ki | 4 | — | |
GMIJWONFGCBOTB
|
7.8 | Ki | 4 | — | |
JVQDBDSYYMHCTL
|
7.8 | Ki | 4 | — | |
KBPQIDCZZMLFSH
|
7.8 | Ki | 4 | — | |
KVHQJEIOEXQVBK
|
7.8 | Ki | 4 | — | |
QGGLESNNYLSYEA
|
7.8 | IC50 | 3 | — | |
TYQILDGWSUOEBL
|
7.8 | Ki | 2 | — | |
TYQILDGWSUOEBL
|
7.8 | Ki | 4 | — | |
SAIXTBXXQWMWMW
|
7.8 | IC50 | 5 | — | |
ZEBTXFXNRXGPKC
|
7.8 | IC50 | 3 | — | |
ZSTCZFASHGPJKC
|
7.8 | Ki | 4 | — | |
AILLCBRMQPBNQN
|
7.8 | IC50 | 13 | — | |
HIDZIHZHRJJHIB
|
7.8 | IC50 | 2 | — | |
HOFGFUOFMADIHI
|
7.8 | IC50 | 3 | — | |
KTCCFGNAPQZORP
|
7.8 | IC50 | 3 | — | |
LGYATYGAQMYTGJ
|
7.8 | IC50 | 2 | — | |
MONFIAJYKZCCDQ
|
7.8 | IC50 | 3 | — | |
NJQPWPCWSTUVSO
|
7.8 | IC50 | 2 | — | |
QWDLZMUWYCLKFF
|
7.8 | IC50 | 10 | — | |
RXMMUXFFAPOLCQ
|
7.8 | IC50 | 3 | — | |
TWZUBEUBTUGWHY
|
7.8 | IC50 | 3 | — | |
USXJKWQIDCWKGZ
|
7.8 | Ki | 10 | — | |
VHWYHHQIYHLXIJ
|
7.8 | IC50 | 2 | — | |
VKMLLLMORNMXCU
|
7.8 | IC50 | 2 | — | |
ZQLILUVVXPRXLE
|
7.8 | IC50 | 3 | — | |
ZVMZOIRSIBVTNJ
|
7.8 | IC50 | 3 | — | |
ZZGZCQUEZVKTAM
|
7.8 | IC50 | 3 | — | |
VZRDHFCDSYWOHQ
|
7.8 | Ki | 4 | — | |
AHJRHEGDXFFMBM
|
7.8 | IC50 | 28 | — | |
AOQGFYCQRQMBKO
|
7.8 | IC50 | 2 | — | |
BAMUDEHGCAVPNN
|
7.8 | IC50 | 2 | — | |
BVQJZQPMZIISOS
|
7.8 | IC50 | 3 | — | |
CMTNNQFGCHCRSZ
|
7.8 | IC50 | 2 | — | |
CXRFVRQTMSLWOK
|
7.8 | IC50 | 4 | — | |
DSYAGVYPTCYGKP
|
7.8 | IC50 | 5 | — | |
FDNONPIMUKKMQB
|
7.8 | IC50 | 2 | — | |
FUHVDXOTJYWTON
|
7.8 | IC50 | 2 | — | |
IYYKYLPYCPFJHV
|
7.8 | IC50 | 2 | — | |
JFFPDPOBHVQORV
|
7.8 | IC50 | 2 | — | |
JLIDFAZKTWWWCN
|
7.8 | IC50 | 5 | — | |
JWNZXWGMBRXMPK
|
7.8 | IC50 | 4 | — |