Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DULGXBOFHQPIOB
|
7.9 | IC50 | 3 | — | |
FRNNWASSAAUPGS
|
7.9 | IC50 | 2 | — | |
LDEHCBTUGDRPFY
|
7.9 | IC50 | 2 | — | |
MLLWORSXSDVTQA
|
7.9 | IC50 | 2 | — | |
PAXKGQZKOJPPEG
|
7.9 | IC50 | 5 | Yes | |
QXFDGSVFDQJMHD
|
7.9 | IC50 | 2 | — | |
RAFUPHSGKSPIHL
|
7.9 | IC50 | 2 | — | |
UQXIOTQQUSBFRU
|
7.9 | IC50 | 3 | — | |
VKWVMZJDIBGOSR
|
7.9 | IC50 | 2 | — | |
VMOLERSXTKLIOK
|
7.9 | IC50 | 3 | — | |
PJNDWVHDRGLRDW
|
7.9 | Ki | 4 | — | |
SQAZXWOTKSSCBZ
|
7.9 | IC50 | 3 | — | |
VXTCGNYHDLHMIV
|
7.9 | IC50 | 2 | — | |
WEIJWGUXTMLFKT
|
7.9 | IC50 | 3 | — | |
WUNBOTQFUIFMPU
|
7.9 | Ki | 4 | — | |
FZXIKXAEEYJOOI
|
7.9 | Ki | 4 | — | |
JEUQWNQSQIEFOJ
|
7.9 | IC50 | 3 | — | |
KGVDWEZLAHTJSJ
|
7.9 | IC50 | 8 | — | |
OUTLYXINOACMSY
|
7.9 | IC50 | 4 | — | |
PBEICQQHXUBGMD
|
7.9 | Ki | 4 | — | |
VKQLKJVYGXNJBA
|
7.9 | Ki | 4 | — | |
BOEVQFOAJBRYBJ
|
7.9 | IC50 | 4 | — | |
CFBGLJFJVCLSNN
|
7.9 | IC50 | 2 | — | |
FJVCRQHDTUXVMH
|
7.9 | Ki | 4 | — | |
GNKARCUXNWYAPQ
|
7.9 | IC50 | 5 | — | |
NRMCNHRZOLZAMB
|
7.9 | IC50 | 2 | — | |
RUYVBOROXISBTA
|
7.9 | IC50 | 2 | — | |
UQVFTDIMDMBMCP
|
7.9 | IC50 | 2 | — | |
VSZKYBBLLRBZLS
|
7.9 | IC50 | 3 | — | |
VTEOJXOIAQEYFO
|
7.9 | Ki | 4 | — | |
WISHLJZJMNBRMX
|
7.9 | IC50 | 9 | — | |
WQIITJQRBLEBPL
|
7.9 | IC50 | 3 | — | |
YTNZPCAMOLEZQS
|
7.9 | IC50 | 2 | — | |
ZIJYDOFMALQXKA
|
7.9 | IC50 | 2 | — | |
CDZRXVMQLQSKPO
|
7.9 | Ki | 3 | — | |
GCZKEPXNHVTKDQ
|
7.9 | Ki | 4 | — | |
HFKMNAUFISJBSK
|
7.9 | IC50 | 6 | — | |
UJHKKNOWOJMKCR
|
7.9 | IC50 | 3 | — | |
UKUVHVSOTZPZBW
|
7.9 | IC50 | 4 | — | |
XNFJUHZLDMOZHP
|
7.9 | IC50 | 2 | — | |
JNCFUVQWIVLATB
|
7.9 | IC50 | 3 | — | |
UOXNTMLLQKBLLA
|
7.9 | IC50 | 4 | — | |
IFXJYXJVOYKBDP
|
7.9 | IC50 | 8 | — | |
NTLJHBLBHSTNJY
|
7.9 | Ki | 4 | — | |
QYJLBHRAPDJOSO
|
7.9 | Ki | 4 | — | |
DHXAFRBSJGTAFK
|
7.8 | IC50 | 3 | — | |
DNFNQGHGGVBVSY
|
7.8 | IC50 | 3 | — | |
HXYNOSRTKCYTLX
|
7.8 | IC50 | 2 | — | |
JGXWHAWACJWVKA
|
7.8 | IC50 | 2 | — | |
JZIDYKXHTRKVEP
|
7.8 | IC50 | 5 | — |