Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TZDIAPGMMCTLTB
|
8.1 | IC50 | 3 | — | |
URMNAIXMQBTMBC
|
8.1 | IC50 | 3 | — | |
ZEIYUGJMJHYICR
|
8.1 | IC50 | 3 | — | |
DHMHGKLKKIGMHX
|
8.1 | IC50 | 3 | — | |
FCFWUBWRSPVMRL
|
8.1 | Ki | 4 | — | |
HZNBZEKLTOCERM
|
8.1 | IC50 | 2 | — | |
UZWDCWONPYILKI
|
8.1 | IC50 | 47 | — | |
PBPBUOMTKKDUEJ
|
8.1 | Ki | 4 | — | |
SROFUFWCKOGJNG
|
8.1 | Ki | 4 | — | |
YOPAUTRVBICJOC
|
8.1 | IC50 | 2 | — | |
APKPENVZICKJOY
|
8.1 | IC50 | 2 | — | |
GMUVHXBIPOWLCK
|
8.1 | IC50 | 3 | — | |
MDSUHMLXNPZZHO
|
8.1 | IC50 | 7 | — | |
QJPGYWGHFLUOIS
|
8.1 | IC50 | 2 | — | |
VQWRERKTQFNERF
|
8.1 | IC50 | 8 | — | |
WSYHYLUWICJSJV
|
8.1 | IC50 | 8 | — | |
AWQCYDKXNFPPQC
|
8.1 | IC50 | 3 | — | |
DXKQFNWEGVJNQT
|
8.1 | IC50 | 2 | — | |
FCYRMRVUDQMNHO
|
8.1 | Ki | 4 | — | |
FMYDWZBWZKJPCK
|
8.1 | IC50 | 4 | — | |
ITDDDMFXMSWPBU
|
8.1 | IC50 | 3 | — | |
NGYRNPFGDZALOR
|
8.1 | IC50 | 3 | — | |
OIQCBGFNCAFMQX
|
8.1 | Ki | 10 | — | |
ONYDIUVHLRZYJB
|
8.1 | IC50 | 3 | — | |
RMYBOOZEFJJYAI
|
8.1 | IC50 | 2 | — | |
VJFMIBISXQANRG
|
8.1 | Ki | 8 | — | |
XIWVBPODMDKKKM
|
8.1 | Ki | 4 | — | |
MMHOKKKPDYDUDS
|
8.0 | Ki | 4 | — | |
SPPKSFFDOAHKJG
|
8.0 | Ki | 4 | — | |
YTFXXQYRDAFPOR
|
8.0 | IC50 | 2 | — | |
ZAPGHPQYYDYEQW
|
8.0 | IC50 | 6 | — | |
ZTEGEMFKBZMGOF
|
8.0 | IC50 | 9 | — | |
LFGOPXAPKINMIT
|
8.0 | Ki | 4 | — | |
QPSCTAMMABVQIH
|
8.0 | IC50 | 3 | — | |
GPJWAQYXKOYKLZ
|
8.0 | IC50 | 2 | — | |
KZVVZDSUJLUKFC
|
8.0 | Ki | 4 | — | |
OFUSTOXZRPWIMF
|
8.0 | Ki | 4 | — | |
DHFGHSZKOLMKGI
|
8.0 | IC50 | 2 | — | |
GPNPQTRGIAJGBJ
|
8.0 | Ki | 4 | — | |
HVGWRZOBPIJOSS
|
8.0 | IC50 | 2 | — | |
LASUSMNDZBNUAS
|
8.0 | Ki | 4 | — | |
BKMZBHQCZLDPLV
|
8.0 | IC50 | 3 | — | |
BWIZOFRKIJFPNB
|
8.0 | IC50 | 2 | — | |
CATPVVCQUODOLN
|
8.0 | IC50 | 8 | — | |
CZUZPLMVIUUOMD
|
8.0 | Ki | 4 | — | |
DPIODVZRGWTHFY
|
8.0 | IC50 | 2 | — | |
GBVXPZRKGCHAIL
|
8.0 | IC50 | 6 | — | |
HPIIKSFGPMWKJM
|
8.0 | IC50 | 5 | — | |
IJPHYTNUHVHWHD
|
8.0 | IC50 | 2 | — | |
IMDAAVXNKFRYNY
|
8.0 | Ki | 10 | — |