Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IBDBTEISIFQPCU
|
8.1 | Ki | 2 | — | |
MCGKCTAGXKRXDO
|
8.1 | Ki | 4 | — | |
MYNSISSWZNWEKP
|
8.1 | IC50 | 2 | — | |
ROMAHJZEHBXJSU
|
8.1 | IC50 | 7 | — | |
HCCNJLKJQAHREN
|
8.1 | IC50 | 3 | — | |
SVXDTIUTCGVODS
|
8.1 | IC50 | 3 | — | |
BMBAGOPVYVYLRK
|
8.1 | IC50 | 3 | — | |
CDJMGTBBCJIMSO
|
8.1 | IC50 | 3 | — | |
CJOCXJOHQLURIU
|
8.1 | IC50 | 5 | — | |
DIEPAOLAVQCUMJ
|
8.1 | IC50 | 3 | — | |
DMINDFPRECTTDS
|
8.1 | IC50 | 3 | — | |
DQBASRYERZQRJJ
|
8.1 | IC50 | 15 | — | |
HLOKDQHOCMHLLI
|
8.1 | IC50 | 7 | — | |
HLZLNALDBVRHFY
|
8.1 | IC50 | 3 | — | |
KPCVCNZJVUSNOC
|
8.1 | IC50 | 5 | — | |
MBYWSZFZJVGHPT
|
8.1 | IC50 | 3 | — | |
MPLKCBASNJCULZ
|
8.1 | IC50 | 3 | — | |
NELAJQKSVYVYHT
|
8.1 | IC50 | 3 | — | |
OIHTZDBVUWNXKY
|
8.1 | IC50 | 3 | — | |
PJJRCQULLSOBAU
|
8.1 | IC50 | 3 | — | |
QHHRSGXUBJPGLM
|
8.1 | IC50 | 3 | — | |
QJBKKUZKLLCQQP
|
8.1 | IC50 | 3 | — | |
STKZFFVPVRFGPN
|
8.1 | IC50 | 3 | — | |
VGMLIUVYQAAPOV
|
8.1 | IC50 | 2 | — | |
WFGZEHUPMAIWSS
|
8.1 | IC50 | 3 | — | |
YKKFCIYOTDLCGD
|
8.1 | Ki | 4 | — | |
ZAFJPCZWYDCVJT
|
8.1 | IC50 | 3 | — | |
ZBSLNLOKLQOETL
|
8.1 | IC50 | 3 | — | |
ZCGJMLAZQFNDAN
|
8.1 | IC50 | 2 | — | |
BBRFMBZEPLRVBF
|
8.1 | Ki | 4 | — | |
DLIDUXYWQPLFEM
|
8.1 | IC50 | 5 | Yes | |
HVTYFANOGPVRAE
|
8.1 | IC50 | 3 | — | |
QSWXQGNVXUPASL
|
8.1 | Ki | 4 | — | |
YJXCLPMUNHAMQF
|
8.1 | Ki | 4 | — | |
AWPNCYPNCSCZFL
|
8.1 | IC50 | 4 | — | |
BBUVDDPUURMFOX
|
8.1 | IC50 | 4 | — | |
CNEMATMUMUNODK
|
8.1 | IC50 | 2 | — | |
DZWLTXLJZHDQOP
|
8.1 | IC50 | 2 | — | |
GKTNOVUFHDVNPA
|
8.1 | IC50 | 4 | — | |
LICJOAWXMPKZSX
|
8.1 | Ki | 10 | — | |
LTAGEPXBKGCCEF
|
8.1 | Ki | 4 | — | |
MJICTPPWZJLGIM
|
8.1 | Ki | 4 | — | |
MPUULNLPAQHDGK
|
8.1 | IC50 | 2 | — | |
MRFIWOQUOAXZDO
|
8.1 | Ki | 5 | — | |
QCALUKUBCRTVRC
|
8.1 | Ki | 4 | — | |
QGSJHTSIQFGZDV
|
8.1 | IC50 | 2 | — | |
QTNFANVRKMXUKB
|
8.1 | IC50 | 3 | — | |
QXLHPZGOJNRMDZ
|
8.1 | IC50 | 2 | — | |
RFAFNLAEMWZQJI
|
8.1 | IC50 | 3 | — | |
SISAEGSKELJSQO
|
8.1 | IC50 | 2 | — |