Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVEBMCRIHHZDFG
|
8.2 | Ki | 8 | — | |
VISMKLIGDLCELE
|
8.2 | IC50 | 3 | — | |
DXSFYOCCBPQCIO
|
8.2 | Ki | 4 | — | |
FZDLLCNNEVTCFF
|
8.2 | Ki | 4 | — | |
GUYDOLZTUBMZKV
|
8.2 | Ki | 4 | — | |
HCAPKVUYVLOOHA
|
8.2 | IC50 | 5 | — | |
IIJWYFPAKYPUIM
|
8.2 | IC50 | 8 | — | |
JAZHDXRHOSJZHB
|
8.2 | IC50 | 3 | — | |
KYMNNSMBWCZWCF
|
8.2 | IC50 | 3 | — | |
SWHALWMKROAPPG
|
8.2 | IC50 | 3 | — | |
XMLANQVRPNNKMS
|
8.2 | IC50 | 2 | — | |
XWWYSAVKDKITGM
|
8.2 | IC50 | 2 | — | |
IIWJISYNHGWLAF
|
8.2 | Ki | 4 | — | |
IUYLNMPIDQAYSG
|
8.2 | IC50 | 7 | — | |
KNRZSSHNVWPHLG
|
8.2 | IC50 | 2 | — | |
KOGSYYDLPNMWFL
|
8.2 | Ki | 4 | — | |
PMCGYDRAUVMLBE
|
8.2 | IC50 | 3 | — | |
QXBRBWDRQIISAT
|
8.2 | IC50 | 6 | — | |
QZCCSLYLFPQDDP
|
8.2 | Ki | 4 | — | |
FICIRDHVWSBGDI
|
8.2 | IC50 | 2 | — | |
HXKORJQOSCRLJP
|
8.2 | IC50 | 5 | — | |
KIQWHSXCLUTZKG
|
8.2 | IC50 | 2 | — | |
NOURLRCLQWYULH
|
8.2 | IC50 | 2 | — | |
QNUFZYZRLJGZJL
|
8.2 | IC50 | 10 | — | |
AQZYUSPIXYHTDI
|
8.2 | Ki | 4 | — | |
DABVJURXDMIZKX
|
8.2 | Ki | 7 | — | |
JXJHPQHLHQTQQI
|
8.2 | IC50 | 15 | — | |
KLYIOUNPTCQBFR
|
8.2 | IC50 | 2 | — | |
OIQZLVBXHSEFQP
|
8.2 | IC50 | 6 | — | |
FIHHRMZWXIZLJV
|
8.2 | Ki | 4 | — | |
KQWXMJOPENRODE
|
8.2 | Ki | 4 | — | |
OFGLKFLIMBZBTK
|
8.2 | IC50 | 2 | — | |
DVAPMYJVUZJNDK
|
8.2 | Ki | 4 | — | |
FCWWBOZXMLGFHI
|
8.2 | IC50 | 2 | — | |
HFYYJLJETVWZJA
|
8.2 | IC50 | 2 | — | |
UQAHWAQRLXARGK
|
8.2 | IC50 | 3 | — | |
AMPDZRFNHCTPTF
|
8.2 | Ki | 10 | — | |
AXTGGTFVALFVDO
|
8.2 | IC50 | 6 | — | |
AZYQVHANOGPVQX
|
8.2 | IC50 | 3 | — | |
DHQTVQLYTCGZPM
|
8.2 | IC50 | 2 | — | |
JDIAYVMOUUKPNK
|
8.2 | IC50 | 5 | — | |
JGXWHAWACJWVKA
|
8.2 | IC50 | 2 | — | |
PFJVPPHRFDWODX
|
8.2 | Ki | 4 | — | |
RATTVJZQLHAPSM
|
8.2 | IC50 | 3 | — | |
VMVGVNIHPKFEIL
|
8.2 | IC50 | 2 | — | |
WZQSDNJOORXCQA
|
8.2 | IC50 | 3 | — | |
XJKXAULUFNXVMK
|
8.2 | Ki | 4 | — | |
XLZANAXESDHDPY
|
8.2 | Ki | 8 | — | |
YZVFJIYEYQIHIP
|
8.2 | IC50 | 15 | — | |
AZENZYQBDCPVQO
|
8.1 | IC50 | 3 | — |