Target Details
| UniProt AC | Q00534 |
|---|---|
| Gene Symbol | CDK6 |
| Protein Name | Cyclin-dependent kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,915
- Clinical molecules 17
- Avg pChEMBL 7.56
KEGG Pathways (23)
- Breast cancer
- Cell cycle
- Cellular senescence
- Chronic myeloid leukemia
- Cushing syndrome
- Epstein-Barr virus infection
- Glioma
- Hepatitis C
- Hepatocellular carcinoma
- Human cytomegalovirus infection
- Human papillomavirus infection
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Measles
- Melanoma
- MicroRNAs in cancer
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (1,915)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORANZZBUKCNAKJ
|
8.3 | IC50 | 2 | — | |
QVWFFHVKVHIONZ
|
8.3 | Ki | 4 | — | |
RKGAIIIRLQHASS
|
8.3 | IC50 | 3 | — | |
UPQKBKLECVIXJR
|
8.3 | IC50 | 12 | — | |
VASFNXBXECJRSY
|
8.3 | IC50 | 15 | — | |
VWXHIFNNYBTKPP
|
8.3 | IC50 | 3 | — | |
VYJDSETVCMXOBL
|
8.3 | Ki | 4 | — | |
BURBSRHEPGFKHA
|
8.3 | IC50 | 2 | — | |
IZSLXRORDBBGDE
|
8.3 | IC50 | 3 | — | |
NEMLRBSGBSXGPB
|
8.3 | Ki | 4 | — | |
OBTPCSNROCZPDN
|
8.3 | IC50 | 2 | — | |
OCCSFFDCCOSIJB
|
8.3 | Ki | 4 | — | |
OVSVIUOGHPWXNH
|
8.3 | IC50 | 6 | — | |
SISAEGSKELJSQO
|
8.3 | IC50 | 2 | — | |
VZPLQNFSKCQLPB
|
8.3 | IC50 | 3 | — | |
ZRBMKKBZXGSURN
|
8.3 | IC50 | 2 | — | |
GSPKCQHHHDAZPV
|
8.3 | Ki | 4 | — | |
OIJRETQRRUTHKW
|
8.3 | IC50 | 2 | — | |
VQPRNWUDMGAWOA
|
8.3 | IC50 | 2 | — | |
YRUAMADPOZOPBF
|
8.3 | IC50 | 7 | — | |
QZILCAFHEDWHIC
|
8.3 | Ki | 4 | — | |
DWVMFMWELQFMNJ
|
8.3 | IC50 | 3 | — | |
GOPDWIWLPUUQTK
|
8.3 | IC50 | 3 | — | |
GYDXFTMHNUETBY
|
8.3 | IC50 | 5 | — | |
SZRLOUJSZUQGCD
|
8.3 | IC50 | 3 | — | |
BWTNWYUWKYKEBW
|
8.2 | Ki | 4 | — | |
JNZTWAOEOYBNNP
|
8.2 | IC50 | 5 | — | |
JUQKGEXKBSXXHM
|
8.2 | IC50 | 2 | — | |
RAIPOUVWZMOUJL
|
8.2 | IC50 | 3 | — | |
UMJDAZSXABEMLH
|
8.2 | IC50 | 4 | — | |
APLCQEOLIQVWQN
|
8.2 | Ki | 4 | — | |
AQSKGIKUFDLXKA
|
8.2 | Ki | 4 | — | |
FIGHMADYPRDXEQ
|
8.2 | IC50 | 6 | — | |
KHUHONPSWMPDIC
|
8.2 | Ki | 4 | — | |
KTAKVDASVPBVHO
|
8.2 | IC50 | 2 | — | |
NOUVQMCOTSOPTN
|
8.2 | IC50 | 2 | — | |
NROJANSVZVKJQE
|
8.2 | IC50 | 2 | — | |
OYDSNFVBFPSPON
|
8.2 | Ki | 4 | — | |
SKRUYIPFBIYOHZ
|
8.2 | IC50 | 2 | — | |
SSIOYGMEKCPFAV
|
8.2 | IC50 | 6 | — | |
USBNWJQZRGQXPN
|
8.2 | IC50 | 3 | — | |
WADAAQHFKRCHPA
|
8.2 | IC50 | 2 | — | |
YVMZPLLKFCKPIL
|
8.2 | IC50 | 2 | — | |
DKTHMZUTCUNQAZ
|
8.2 | IC50 | 5 | — | |
IQHJQQIVUNNQTR
|
8.2 | Ki | 4 | — | |
UEGPMXKTKCKXOK
|
8.2 | IC50 | 3 | — | |
XMWHZKQZVIMLTH
|
8.2 | IC50 | 2 | — | |
BXSSOAIGLMVYQR
|
8.2 | Ki | 8 | — | |
HFMQOFFEBHLBLK
|
8.2 | IC50 | 3 | — | |
KPEABKWUJCTBRM
|
8.2 | IC50 | 5 | — |