Target Details
| UniProt AC | Q00526 |
|---|---|
| Gene Symbol | CDK3 |
| Protein Name | Cyclin-dependent kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 152
- Clinical molecules 10
- Avg pChEMBL 7.09
Active Molecules (152)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BDLBLCWMNJLLLI
|
7.3 | IC50 | 5 | — | |
NBSJZWFDNFWQDN
|
7.3 | IC50 | 29 | — | |
ICVWYIZCPUIPOY
|
7.3 | IC50 | 7 | — | |
UBGXMRPQIYVDEN
|
7.3 | IC50 | 4 | — | |
OUSFTKFNBAZUKL
|
7.2 | Kd | 58 | Yes | |
CELCCCWTAADGDV
|
7.2 | IC50 | 15 | — | |
NKSJUACUARPPLH
|
7.2 | IC50 | 13 | — | |
YQOZFMRCEONJEU
|
7.2 | IC50 | 13 | — | |
UCVRLTXXBKZAOV
|
7.2 | IC50 | 5 | — | |
PGETVCQNSNDKAY
|
7.2 | IC50 | 6 | — | |
OVBAFUGPHNUQFH
|
7.2 | IC50 | 7 | — | |
YCWRVLHIXKSYQM
|
7.2 | IC50 | 5 | — | |
SMWJYKRUKGMKJV
|
7.1 | IC50 | 11 | — | |
XNLQUWXXCRJCDC
|
7.1 | IC50 | 4 | — | |
ZPHBEDTYTQWLFC
|
7.1 | IC50 | 13 | — | |
RPGZQOOZHIEPJW
|
7.1 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.1 | Kd | 18 | — | |
UWZBUGMYQWUJLU
|
7.1 | IC50 | 5 | — | |
ODPGGGTTYSGTGO
|
7.1 | Kd | 153 | — | |
YJJUWEQVCJXIPR
|
7.1 | IC50 | 5 | — | |
AKIBGBJFUGFCIJ
|
7.1 | IC50 | 7 | — | |
MXKWVQJXDBWLPO
|
7.1 | IC50 | 6 | — | |
WYHDWGBEHMLGBC
|
7.1 | IC50 | 3 | — | |
YPSCKJWJIXZMSC
|
7.0 | IC50 | 15 | — | |
ATBAETXFFCOZOY
|
7.0 | IC50 | 39 | — | |
JZQPZFUOGWPPOG
|
7.0 | IC50 | 6 | — | |
AJPNQVZYWOGOKN
|
7.0 | IC50 | 5 | — | |
NUBBIJVOSXWZTF
|
7.0 | IC50 | 13 | — | |
RUQCKUPFMSPOOF
|
7.0 | IC50 | 3 | — | |
YBLPMNNVXVEMKC
|
7.0 | IC50 | 5 | — | |
CEIJSVLEARLWRF
|
7.0 | IC50 | 13 | — | |
JNYWLVWHCGXRPJ
|
7.0 | IC50 | 4 | — | |
ZLNVBIGZYRPQKY
|
6.9 | IC50 | 15 | — | |
GSYUZRLLPWNNAL
|
6.9 | IC50 | 6 | — | |
PUELPOFWJXDUSU
|
6.9 | IC50 | 4 | — | |
LTDFDPHSEHTUCI
|
6.9 | IC50 | 5 | — | |
ODBLPALGDXNFKK
|
6.9 | IC50 | 4 | — | |
OZZGCHZTKBHAMX
|
6.9 | IC50 | 4 | — | |
ZLPVQTFOPHTMQK
|
6.9 | IC50 | 4 | — | |
ULMMSSXMAQOVME
|
6.9 | IC50 | 7 | — | |
ZCCPLJOKGAACRT
|
6.9 | Kd | 599 | — | |
IAYGCINLNONXHY
|
6.9 | Kd | 50 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
QILDHEURHSGJQY
|
6.8 | IC50 | 3 | — | |
XKPQEHCOXUTCAV
|
6.8 | IC50 | 4 | — | |
ZFWMAWDMXORLSP
|
6.8 | IC50 | 6 | — | |
RSRKFXROJZFOAM
|
6.8 | IC50 | 3 | — | |
ISBMMEQKVMLOCZ
|
6.8 | IC50 | 3 | — | |
QTMWJQCPEOTFSB
|
6.8 | IC50 | 5 | — | |
JIUQQBHMLCPYSQ
|
6.8 | IC50 | 3 | — |