Target Details
| UniProt AC | Q00526 |
|---|---|
| Gene Symbol | CDK3 |
| Protein Name | Cyclin-dependent kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 152
- Clinical molecules 10
- Avg pChEMBL 7.09
Active Molecules (152)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQHPGIWKYQJUIE
|
9.2 | IC50 | 7 | — | |
DQBASRYERZQRJJ
|
9.0 | IC50 | 15 | — | |
XLSYZSRXVVCHLS
|
8.7 | IC50 | 48 | — | |
IAPISFUJUUDVNW
|
8.6 | IC50 | 15 | — | |
JRNJNYBQQYBCLE
|
8.5 | Kd | 40 | Yes | |
YLWSVZLNZZVTSM
|
8.3 | IC50 | 15 | — | |
FMUUGBFOPCVEBP
|
8.2 | IC50 | 7 | — | |
BKCOGSHTNWTZNI
|
8.2 | IC50 | 15 | — | |
FKAJEPVSQITQLJ
|
8.2 | IC50 | 15 | — | |
UELYDGOOJPRWGF
|
8.2 | IC50 | 13 | — | |
HKSZLNNOFSGOKW
|
8.2 | IC50 | 408 | — | |
HUXYBQXJVXOMKX
|
8.1 | Kd | 28 | — | |
VXBAJLGYBMTJCY
|
8.1 | IC50 | 34 | Yes | |
YZVFJIYEYQIHIP
|
8.1 | IC50 | 15 | — | |
PEJLZSHWCASCSY
|
8.1 | IC50 | 6 | — | |
KGJVKYSVVOQPDL
|
8.0 | IC50 | 13 | — | |
KJHOORCYJSBANN
|
8.0 | IC50 | 15 | — | |
VASFNXBXECJRSY
|
8.0 | IC50 | 15 | — | |
RVKNONNXSNALJV
|
8.0 | IC50 | 21 | — | |
LEHFYLKYODNMCD
|
7.9 | IC50 | 5 | — | |
SFFYJMOAIFNGCJ
|
7.9 | IC50 | 6 | — | |
RWSCYFXGWJPUQX
|
7.9 | IC50 | 15 | — | |
QZCITBQFXYREEJ
|
7.8 | IC50 | 7 | — | |
FKAJEPVSQITQLJ
|
7.8 | IC50 | 15 | — | |
JTIFUJUJDWUQEV
|
7.7 | IC50 | 12 | — | |
GAPTWFVBSQIGOP
|
7.7 | IC50 | 6 | — | |
FNAWEKRTBLXUJI
|
7.7 | IC50 | 7 | — | |
AVIWDYSJSPOOAR
|
7.6 | IC50 | 11 | — | |
ITHPWIHYZQLUIG
|
7.6 | IC50 | 7 | — | |
PHZDWQYTFQOSSZ
|
7.6 | IC50 | 15 | — | |
TYSWNLQZLBRNSE
|
7.6 | IC50 | 15 | — | |
XQKRWDLELRIZOC
|
7.6 | IC50 | 7 | — | |
CXMKIWPGGSLHRE
|
7.5 | IC50 | 15 | — | |
FJXAKWGPTCSFIG
|
7.5 | IC50 | 7 | — | |
FLIVKVQMXOAQAK
|
7.5 | IC50 | 15 | — | |
PFRMQZGBTCACGO
|
7.5 | IC50 | 7 | — | |
PXKQKKHBHPRTEG
|
7.5 | IC50 | 6 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
VGAKNPKNIZJLEF
|
7.5 | IC50 | 6 | — | |
KOZFSFOOLUUIGY
|
7.5 | Kd | 88 | Yes | |
RAOPEUTYHRNFHJ
|
7.5 | IC50 | 7 | — | |
ZJKDYTFNXUBLEQ
|
7.5 | IC50 | 15 | — | |
FVEIPMUKOTZXBA
|
7.4 | IC50 | 7 | — | |
JXJHPQHLHQTQQI
|
7.4 | IC50 | 15 | — | |
WOBKYDKXSVLQGJ
|
7.4 | IC50 | 7 | — | |
FHDYRKMYVDZJBI
|
7.4 | IC50 | 6 | — | |
ZODPLLYTMWNTCA
|
7.4 | IC50 | 7 | — | |
MLCHXEPEMWHPKH
|
7.3 | IC50 | 7 | — | |
JCAKIRPULCVXNW
|
7.3 | IC50 | 6 | — | |
SGOFJRIGAKFXAH
|
7.3 | IC50 | 6 | — |