Target Details
| UniProt AC | P9WI81 |
|---|---|
| Gene Symbol | pknB |
| Protein Name | Serine/threonine-protein kinase PknB |
| Organism | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03793 (PASTA) PF00069 (Pkinase) |
Summary
- Multi-target molecules 18
- Clinical molecules 5
- Avg pChEMBL 7.37
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KGPGFQWBCSZGEL
|
8.5 | Kd | 59 | Yes | |
XZXHXSATPCNXJR
|
8.4 | Kd | 165 | Yes | |
JOLXSDWLLOKVDT
|
8.4 | Ki | 2 | — | |
RQBXIYXQKQNKEN
|
8.4 | Ki | 4 | — | |
XUQQFBJTQJYWPD
|
7.6 | Ki | 2 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
BKVJIBAADPVALB
|
7.4 | Ki | 5 | — | |
UHNFOKVJWUABIX
|
7.3 | Ki | 5 | — | |
UASKPELCJPQDEL
|
7.3 | Ki | 4 | — | |
UIARLYUEJFELEN
|
7.3 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 408 | — | |
KCPRSPILMCRMSU
|
7.1 | Ki | 5 | — | |
WINHZLLDWRZWRT
|
7.1 | Kd | 201 | Yes | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
GUBJNPWVIUFSTR
|
6.8 | Kd | 103 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
PIQCTGMSNWUMAF
|
6.5 | Kd | 137 | Yes | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — |