Target Details
| UniProt AC | P9WFK7 |
|---|---|
| Gene Symbol | eis |
| Protein Name | N-acetyltransferase Eis |
| Organism | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF17668 (Acetyltransf_17) PF13527 (Acetyltransf_9) PF13530 (SCP2_2) |
Summary
- Multi-target molecules 5
- Clinical molecules 1
- Avg pChEMBL 6.25
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKLNONIVDFXQRX
|
6.5 | IC50 | 4 | — | |
LNEPOXFFQSENCJ
|
6.4 | IC50 | 33 | Yes | |
ZNOLNAPJKOYTHY
|
6.2 | IC50 | 2 | — | |
XDFPJEPCZSJPQC
|
6.1 | IC50 | 2 | — | |
FEFFZKPQSVTBAY
|
6.1 | IC50 | 2 | — |