Target Details
| UniProt AC | P98161 |
|---|---|
| Gene Symbol | PKD1 |
| Protein Name | Polycystin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00059 (Lectin_C) PF13855 (LRR_8) PF00801 (PKD) PF08016 (PKD_channel) PF01477 (PLAT) PF20519 (Polycystin_dom) PF02010 (REJ) PF01822 (WSC) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 7.59
Associated Diseases (1)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JAMGGIDPOXFRAM
|
9.5 | Ki | 3 | — | |
SUQYTYOVPXAUGB
|
9.3 | Ki | 3 | — | |
BOJKFRKNLSCGHY
|
7.9 | Ki | 3 | — | |
CPXHOALOZNWMML
|
7.8 | Ki | 3 | — | |
LUZOFMGZMUZSSK
|
7.4 | Ki | 3 | — | |
LVLFSSZNAIKYCD
|
7.1 | IC50 | 19 | — | |
BGFPMEIULZPARM
|
7.0 | Ki | 3 | — | |
GMAWUPHGBKLOEK
|
6.9 | IC50 | 2 | — | |
LQSHXYHWYGKAMX
|
6.9 | IC50 | 2 | — | |
PWTCCMJTPHCGMS
|
6.8 | Ki | 3 | — | |
QRHDTFFVGFIUKH
|
6.8 | IC50 | 3 | — |